MiR-146a-5p-enriched exosomes inhibit M1 macrophage activation and inflammatory response by targeting CD80

Mol Biol Rep. 2024 Nov 8;51(1):1133. doi: 10.1007/s11033-024-10088-5.

Abstract

Background: Previous studies have demonstrated that miR-146a-5p negatively regulated the intrinsic immune and inflammatory responses, whether the miR-146a-5p-enriched exosomes possess the anti-inflammation effect remains unclear. This study aimed to investigate the effect of miR-146a-5p-enriched exosomes on M1 macrophage activation and inflammatory response and the potential molecular mechanism.

Methods: GEO database was used to analyze the expression of miR-146a-5p in serum exosomes of MASH patients. MiR-146a-5p levels in primary hepatocytes, macrophages, and serum exosomes of MASH mice were measured. MiR-146a-5p-enriched exosomes were constructed and the effects on M1 macrophages activation and inflammatory factors release were investigated. The target gene of miR-146a-5p was predicted and verified.

Results: Serum exosomal miR-146a-5p level was decreased in MASH patients analyzed by GEO database. The miR-146a-5p levels in primary cultured hepatocytes and macrophages of MASH mice were decreased. Serum exosomal miR-146a-5p level was decreased and negatively correlated with the concentrations of IL-6 in MASH mice. Furthermore, miR-146a-5p-enriched exosomes inhibited the M1 macrophages activation and the expression of pro-inflammatory factors MCP-1, IL-6, and TNF-α. CD80 was predicted as the potential target gene of miR-146a-5p, and the expression of CD80 was regulated by miR-146a-5p. In addition, the inhibitory effect of miR-146a-5p on M1 macrophages activation and inflammatory factors release was restored when CD80 was over-expressed.

Conclusions: This study demonstrated that miR-146a-5p-enriched exosomes can inhibit the M1 macrophages activation and reduce the release of pro-inflammatory factors by targeting CD80.

Keywords: CD80; Exosome; Metabolic dysfunction-associated steatohepatitis; MiR-146a-5p.

MeSH terms

  • Animals
  • B7-1 Antigen* / genetics
  • B7-1 Antigen* / metabolism
  • Exosomes* / genetics
  • Exosomes* / metabolism
  • Hepatocytes / metabolism
  • Humans
  • Inflammation* / genetics
  • Inflammation* / metabolism
  • Interleukin-6 / genetics
  • Interleukin-6 / metabolism
  • Macrophage Activation* / genetics
  • Macrophages* / immunology
  • Macrophages* / metabolism
  • Male
  • Mice
  • MicroRNAs* / genetics
  • MicroRNAs* / metabolism
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • MicroRNAs
  • MIRN146 microRNA, human
  • Mirn146 microRNA, mouse
  • B7-1 Antigen
  • Interleukin-6
  • Tumor Necrosis Factor-alpha