HHSN271200800025C/MH/NIMH NIH HHS/United States[Grants and Funding] - Search Results

Year	Number of Results
2012	3
2013	3
2014	1
2016	5
2017	1
2018	1
2019	3
2020	5
2021	2
2022	4
2023	3
2024	0

1

Structure of a Hallucinogen-Activated Gq-Coupled 5-HT_2A Serotonin Receptor.

Kim K, Che T, Panova O, DiBerto JF, Lyu J, Krumm BE, Wacker D, Robertson MJ, Seven AB, Nichols DE, Shoichet BK, Skiniotis G, Roth BL. Kim K, et al. Cell. 2020 Sep 17;182(6):1574-1588.e19. doi: 10.1016/j.cell.2020.08.024. Cell. 2020. PMID: 32946782 Free PMC article.

2

Discovery of G Protein-Biased Antagonists against 5-HT₇R.

Kwag R, Lee J, Kim D, Lee H, Yeom M, Woo J, Cho Y, Kim HJ, Kim J, Keum G, Jeon B, Choo H. Kwag R, et al. J Med Chem. 2021 Sep 23;64(18):13766-13779. doi: 10.1021/acs.jmedchem.1c01093. Epub 2021 Sep 14. J Med Chem. 2021. PMID: 34519505

3

Pharmacosynthetics: Reimagining the pharmacogenetic approach.

Farrell MS, Roth BL. Farrell MS, et al. Brain Res. 2013 May 20;1511:6-20. doi: 10.1016/j.brainres.2012.09.043. Epub 2012 Oct 9. Brain Res. 2013. PMID: 23063887 Free PMC article. Review.

4

Structure-Activity Studies of 1H-Imidazo[4,5-c]quinolin-4-amine Derivatives as A₃ Adenosine Receptor Positive Allosteric Modulators.

Fallot LB, Suresh RR, Fisher CL, Salmaso V, O'Connor RD, Kaufman N, Gao ZG, Auchampach JA, Jacobson KA. Fallot LB, et al. J Med Chem. 2022 Nov 24;65(22):15238-15262. doi: 10.1021/acs.jmedchem.2c01170. Epub 2022 Nov 11. J Med Chem. 2022. PMID: 36367749 Free PMC article.

5

Specific inhibition of an anticancer target, polo-like kinase 1, by allosterically dismantling its mechanism of substrate recognition.

Park JE, Kirsch K, Lee H, Oliva P, Ahn JI, Ravishankar H, Zeng Y, Fox SD, Kirby SA, Badhwar P, Andresson T, Jacobson KA, Lee KS. Park JE, et al. Proc Natl Acad Sci U S A. 2023 Aug 29;120(35):e2305037120. doi: 10.1073/pnas.2305037120. Epub 2023 Aug 21. Proc Natl Acad Sci U S A. 2023. PMID: 37603740 Free PMC article.

6

Structure activity relationship of novel antiviral nucleosides against Enterovirus A71.

Tosh DK, Toti KS, Hurst BL, Julander JG, Jacobson KA. Tosh DK, et al. Bioorg Med Chem Lett. 2020 Dec 1;30(23):127599. doi: 10.1016/j.bmcl.2020.127599. Epub 2020 Oct 5. Bioorg Med Chem Lett. 2020. PMID: 33031923 Free PMC article.

7

Alicyclic Ring Size Variation of 4-Phenyl-2-naphthoic Acid Derivatives as P2Y₁₄ Receptor Antagonists.

Wen Z, Pramanik A, Lewicki SA, Jung YH, Gao ZG, Randle JCR, Cronin C, Chen Z, Giancotti LA, Whitehead GS, Liang BT, Breton S, Salvemini D, Cook DN, Jacobson KA. Wen Z, et al. J Med Chem. 2023 Jul 13;66(13):9076-9094. doi: 10.1021/acs.jmedchem.3c00664. Epub 2023 Jun 29. J Med Chem. 2023. PMID: 37382926 Free PMC article.

8

New halogenated tris-(phenylalkyl)amines as h5-HT2B receptor ligands.

Kapadia N, Ahmed S, Harding WW. Kapadia N, et al. Bioorg Med Chem Lett. 2016 Jul 15;26(14):3216-3219. doi: 10.1016/j.bmcl.2016.05.079. Epub 2016 May 28. Bioorg Med Chem Lett. 2016. PMID: 27261181

9

Synthesis and pharmacological characterization of multiply substituted 2H-chromene derivatives as P2Y₆ receptor antagonists.

Jung YH, Shah Q, Lewicki SA, Pramanik A, Gopinatth V, Pelletier J, Sévigny J, Iqbal J, Jacobson KA. Jung YH, et al. Bioorg Med Chem Lett. 2022 Nov 1;75:128981. doi: 10.1016/j.bmcl.2022.128981. Epub 2022 Sep 8. Bioorg Med Chem Lett. 2022. PMID: 36089113 Free PMC article.

10

Further studies on C2'-substituted 1-phenylbenzazepines as dopamine D1 receptor ligands.

Giri R, Namballa HK, Sarker A, Alberts I, Harding WW. Giri R, et al. Bioorg Chem. 2022 Oct;127:105953. doi: 10.1016/j.bioorg.2022.105953. Epub 2022 Jun 22. Bioorg Chem. 2022. PMID: 35772367

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