Balzarini J - Search Results

1

1,2,3-Triazole-[2',5'-bis-O-(tert-butyldimethylsilyl)-beta-D- ribofuranosyl]-3'-spiro-5"-(4"-amino-1",2"-oxathiole 2",2"-dioxide) (TSAO) analogues: synthesis and anti-HIV-1 activity.

Alvarez R, Velázquez S, San-Félix A, Aquaro S, De Clercq E, Perno CF, Karlsson A, Balzarini J, Camarasa MJ. Alvarez R, et al. Among authors: balzarini j. J Med Chem. 1994 Nov 25;37(24):4185-94. doi: 10.1021/jm00050a015. J Med Chem. 1994. PMID: 7527463

2

Synthesis of 3' '-substituted TSAO derivatives with anti-HIV-1 and anti-HIV-2 activity through an efficient palladium-catalyzed cross-coupling approach.

Lobatón E, Rodríguez-Barrios F, Gago F, Pérez-Pérez MJ, De Clercq E, Balzarini J, Camarasa MJ, Velázquez S. Lobatón E, et al. Among authors: balzarini j. J Med Chem. 2002 Aug 29;45(18):3934-45. doi: 10.1021/jm020820h. J Med Chem. 2002. PMID: 12190315

3

Acyclic nucleoside analogues as novel inhibitors of human mitochondrial thymidine kinase.

Hernández AI, Balzarini J, Karlsson A, Camarasa MJ, Pérez-Pérez MJ. Hernández AI, et al. Among authors: balzarini j. J Med Chem. 2002 Sep 12;45(19):4254-63. doi: 10.1021/jm011128+. J Med Chem. 2002. PMID: 12213066

4

Improving the selectivity of acyclic nucleoside analogues as inhibitors of human mitochondrial thymidine kinase: replacement of a triphenylmethoxy moiety with substituted amines and carboxamides.

Hernández AI, Balzarini J, Rodríguez-Barrios F, San-Félix A, Karlsson A, Gago F, Camarasa MJ, Pérez-Pérez MJ. Hernández AI, et al. Among authors: balzarini j. Bioorg Med Chem Lett. 2003 Sep 15;13(18):3027-30. doi: 10.1016/s0960-894x(03)00639-5. Bioorg Med Chem Lett. 2003. PMID: 12941326

5

N-3 substituted TSAO derivatives as a probe to explore the dimeric interface of HIV-1 reverse transcriptase.

Bonache MC, Chamorro C, Velázquez S, De Clercq E, Balzarini J, Camarasa MJ, San-Félix A. Bonache MC, et al. Among authors: balzarini j. Nucleosides Nucleotides Nucleic Acids. 2003 May-Aug;22(5-8):947-9. doi: 10.1081/NCN-120022692. Nucleosides Nucleotides Nucleic Acids. 2003. PMID: 14565318 No abstract available.

6

Unusual lability of 5'-O-tert-butyldimethylsilyl group on 4''-acyl TSAO derivatives.

de Castro S, Pérez-Pérez MJ, Lobatón E, De Clercq E, Balzarini J, Camarasa MJ, Velázquez S. de Castro S, et al. Among authors: balzarini j. Nucleosides Nucleotides Nucleic Acids. 2003 May-Aug;22(5-8):959-61. doi: 10.1081/NCN-120022695. Nucleosides Nucleotides Nucleic Acids. 2003. PMID: 14565321 No abstract available.

7

Structure-activity relationship studies on a novel family of specific HIV-1 reverse transcriptase inhibitors.

Bonache MC, Chamorro C, Lobatón E, De Clercq E, Balzarini J, Velázquez S, Camarasa MJ, San-Félix A. Bonache MC, et al. Among authors: balzarini j. Antivir Chem Chemother. 2003 Sep;14(5):249-62. doi: 10.1177/095632020301400504. Antivir Chem Chemother. 2003. PMID: 14694988 Free article.

8

TSAO compounds: the comprehensive story of a unique family of HIV-1 specific inhibitors of reverse transcriptase.

Camarasa MJ, San-Félix A, Velázquez S, Pérez-Pérez MJ, Gago F, Balzarini J. Camarasa MJ, et al. Among authors: balzarini j. Curr Top Med Chem. 2004;4(9):945-63. doi: 10.2174/1568026043388600. Curr Top Med Chem. 2004. PMID: 15134550 Free article. Review.

9

Hybrids of [TSAO-T]-[foscarnet]: The first conjugate of foscarnet with a non-nucleoside reverse transcriptase inhibitor through a labile covalent ester bond.

Velázquez S, Lobatón E, De Clercq E, Koontz DL, Mellors JW, Balzarini J, Camarasa MJ. Velázquez S, et al. Among authors: balzarini j. J Med Chem. 2004 Jun 17;47(13):3418-26. doi: 10.1021/jm031045o. J Med Chem. 2004. PMID: 15189038

10

Synthesis and evaluation of thymine-derived carboxamides against mitochondrial thymidine kinase (TK-2) and related enzymes.

Priego EM, Balzarini J, Karlsson A, Camarasa MJ, Pérez-Pérez MJ. Priego EM, et al. Among authors: balzarini j. Bioorg Med Chem. 2004 Oct 1;12(19):5079-90. doi: 10.1016/j.bmc.2004.07.036. Bioorg Med Chem. 2004. PMID: 15351391

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