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Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors.
Boby ML, Fearon D, Ferla M, Filep M, Koekemoer L, Robinson MC; COVID Moonshot Consortium‡; Chodera JD, Lee AA, London N, von Delft A, von Delft F, Achdout H, Aimon A, Alonzi DS, Arbon R, Aschenbrenner JC, Balcomb BH, Bar-David E, Barr H, Ben-Shmuel A, Bennett J, Bilenko VA, Borden B, Boulet P, Bowman GR, Brewitz L, Brun J, Bvnbs S, Calmiano M, Carbery A, Carney DW, Cattermole E, Chang E, Chernyshenko E, Clyde A, Coffland JE, Cohen G, Cole JC, Contini A, Cox L, Croll TI, Cvitkovic M, De Jonghe S, Dias A, Donckers K, Dotson DL, Douangamath A, Duberstein S, Dudgeon T, Dunnett LE, Eastman P, Erez N, Eyermann CJ, Fairhead M, Fate G, Fedorov O, Fernandes RS, Ferrins L, Foster R, Foster H, Fraisse L, Gabizon R, García-Sastre A, Gawriljuk VO, Gehrtz P, Gileadi C, Giroud C, Glass WG, Glen RC, Glinert I, Godoy AS, Gorichko M, Gorrie-Stone T, Griffen EJ, Haneef A, Hassell Hart S, Heer J, Henry M, Hill M, Horrell S, Huang QYJ, Huliak VD, Hurley MFD, Israely T, Jajack A, Jansen J, Jnoff E, Jochmans D, John T, Kaminow B, Kang L, Kantsadi AL, Kenny PW, Kiappes JL, Kinakh SO, Kovar B, Krojer T, La VNT, Laghnimi-Hahn S, Lefker BA, Levy H, Lithgo RM, Logvinenko IG, Lukacik P, Macdonald HB, MacLean … See abstract for full author list ➔ Boby ML, et al. Among authors: saar k. Science. 2023 Nov 10;382(6671):eabo7201. doi: 10.1126/science.abo7201. Epub 2023 Nov 10. Science. 2023. PMID: 37943932 Free PMC article.
Single-molecule digital sizing of proteins in solution.
Krainer G, Jacquat RPB, Schneider MM, Welsh TJ, Fan J, Peter QAE, Andrzejewska EA, Šneiderienė G, Czekalska MA, Ausserwoeger H, Chai L, Arter WE, Saar KL, Herling TW, Franzmann TM, Kosmoliaptsis V, Alberti S, Hartl FU, Lee SF, Knowles TPJ. Krainer G, et al. Among authors: saar kl. Nat Commun. 2024 Sep 4;15(1):7740. doi: 10.1038/s41467-024-50825-9. Nat Commun. 2024. PMID: 39231922 Free PMC article.
α-Synuclein Oligomers Displace Monomeric α-Synuclein from Lipid Membranes.
Šneiderienė G, Czekalska MA, Xu CK, Jayaram AK, Krainer G, Arter WE, Peter QAE, Castellana-Cruz M, Saar KL, Levin A, Mueller T, Fiedler S, Devenish SRA, Fiegler H, Kumita JR, Knowles TPJ. Šneiderienė G, et al. Among authors: saar kl. ACS Nano. 2024 Jul 9;18(27):17469-17482. doi: 10.1021/acsnano.3c10889. Epub 2024 Jun 25. ACS Nano. 2024. PMID: 38916260 Free PMC article.
Multiomic analyses uncover immunological signatures in acute and chronic coronary syndromes.
Pekayvaz K, Losert C, Knottenberg V, Gold C, van Blokland IV, Oelen R, Groot HE, Benjamins JW, Brambs S, Kaiser R, Gottschlich A, Hoffmann GV, Eivers L, Martinez-Navarro A, Bruns N, Stiller S, Akgöl S, Yue K, Polewka V, Escaig R, Joppich M, Janjic A, Popp O, Kobold S, Petzold T, Zimmer R, Enard W, Saar K, Mertins P, Huebner N, van der Harst P, Franke LH, van der Wijst MGP, Massberg S, Heinig M, Nicolai L, Stark K. Pekayvaz K, et al. Among authors: saar k. Nat Med. 2024 Jun;30(6):1696-1710. doi: 10.1038/s41591-024-02953-4. Epub 2024 May 21. Nat Med. 2024. PMID: 38773340 Free PMC article.
Endothelial Overexpression of TGF-β-Induced Protein Impairs Venous Thrombus Resolution: Possible Role in CTEPH.
Bochenek ML, Saar K, Nazari-Jahantigh M, Gogiraju R, Wiedenroth CB, Münzel T, Mayer E, Fink L, Schober A, Hübner N, Guth S, Konstantinides S, Schäfer K. Bochenek ML, et al. Among authors: saar k. JACC Basic Transl Sci. 2023 Oct 25;9(1):100-116. doi: 10.1016/j.jacbts.2023.08.005. eCollection 2024 Jan. JACC Basic Transl Sci. 2023. PMID: 38362348 Free PMC article.
Targeting the tissue factor coagulation initiation complex prevents antiphospholipid antibody development.
Müller-Calleja N, Grunz K, Nguyen TS, Posma J, Pedrosa D, Meineck M, Hollerbach A, Braun J, Muth S, Schild H, Saar K, Hübner N, Krishnaswamy S, Royce J, Teyton L, Lemmermann N, Weinmann-Menke J, Lackner KJ, Ruf W. Müller-Calleja N, et al. Among authors: saar k. Blood. 2024 Mar 21;143(12):1167-1180. doi: 10.1182/blood.2023022276. Blood. 2024. PMID: 38142429
Theoretical and Data-Driven Approaches for Biomolecular Condensates.
Saar KL, Qian D, Good LL, Morgunov AS, Collepardo-Guevara R, Best RB, Knowles TPJ. Saar KL, et al. Chem Rev. 2023 Jul 26;123(14):8988-9009. doi: 10.1021/acs.chemrev.2c00586. Epub 2023 May 12. Chem Rev. 2023. PMID: 37171907 Free PMC article. Review.
157 results