Conservation of coactivator engagement mechanism enables small-molecule allosteric modulators.
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Proc Natl Acad Sci U S A. 2018 Sep 4;115(36):8960-8965. doi: 10.1073/pnas.1806202115. Epub 2018 Aug 20.
Proc Natl Acad Sci U S A. 2018.
PMID: 30127017
Free PMC article.