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Page 1
Structure-Based Optimization Strategies for G Protein-Coupled Receptor (GPCR) Allosteric Modulators: A Case Study from Analyses of New Metabotropic Glutamate Receptor 5 (mGlu5) X-ray Structures.
Christopher JA, Orgován Z, Congreve M, Doré AS, Errey JC, Marshall FH, Mason JS, Okrasa K, Rucktooa P, Serrano-Vega MJ, Ferenczy GG, Keserű GM. Christopher JA, et al. Among authors: keseru gm. J Med Chem. 2019 Jan 10;62(1):207-222. doi: 10.1021/acs.jmedchem.7b01722. Epub 2018 Mar 1. J Med Chem. 2019. PMID: 29455526
Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs.
Wágner G, Wéber C, Nyéki O, Nógrádi K, Bielik A, Molnár L, Bobok A, Horváth A, Kiss B, Kolok S, Nagy J, Kurkó D, Gál K, Greiner I, Szombathelyi Z, Keseru GM, Domány G. Wágner G, et al. Among authors: keseru gm. Bioorg Med Chem Lett. 2010 Jun 15;20(12):3737-41. doi: 10.1016/j.bmcl.2010.04.075. Epub 2010 Apr 22. Bioorg Med Chem Lett. 2010. PMID: 20483612
Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists.
Galambos J, Wágner G, Nógrádi K, Bielik A, Molnár L, Bobok A, Horváth A, Kiss B, Kolok S, Nagy J, Kurkó D, Bakk ML, Vastag M, Sághy K, Gyertyán I, Gál K, Greiner I, Szombathelyi Z, Keseru GM, Domány G. Galambos J, et al. Among authors: keseru gm. Bioorg Med Chem Lett. 2010 Aug 1;20(15):4371-5. doi: 10.1016/j.bmcl.2010.06.075. Epub 2010 Jun 17. Bioorg Med Chem Lett. 2010. PMID: 20615697
Enthalpic efficiency of ligand binding.
Ferenczy GG, Keseru GM. Ferenczy GG, et al. Among authors: keseru gm. J Chem Inf Model. 2010 Sep 27;50(9):1536-41. doi: 10.1021/ci100125a. J Chem Inf Model. 2010. PMID: 20684566
Thermodynamics guided lead discovery and optimization.
Ferenczy GG, Keserũ GM. Ferenczy GG, et al. Among authors: keseru gm. Drug Discov Today. 2010 Nov;15(21-22):919-32. doi: 10.1016/j.drudis.2010.08.013. Epub 2010 Aug 27. Drug Discov Today. 2010. PMID: 20801227 Review.
Thermodynamics of fragment binding.
Ferenczy GG, Keserű GM. Ferenczy GG, et al. Among authors: keseru gm. J Chem Inf Model. 2012 Apr 23;52(4):1039-45. doi: 10.1021/ci200608b. Epub 2012 Apr 9. J Chem Inf Model. 2012. PMID: 22458364
234 results