Simões-Pires C - Search Results

1

Cross metathesis with hydroxamate and benzamide BOC-protected alkenes to access HDAC inhibitors and their biological evaluation highlighted intrinsic activity of BOC-protected dihydroxamates.

Zwick V, Nurisso A, Simões-Pires C, Bouchet S, Martinet N, Lehotzky A, Ovadi J, Cuendet M, Blanquart C, Bertrand P. Zwick V, et al. Bioorg Med Chem Lett. 2016 Jan 1;26(1):154-9. doi: 10.1016/j.bmcl.2015.11.011. Epub 2015 Nov 11. Bioorg Med Chem Lett. 2016. PMID: 26611919

2

Biphenyl-4-yl-acrylohydroxamic acids: Identification of a novel indolyl-substituted HDAC inhibitor with antitumor activity.

Cincinelli R, Zwick V, Musso L, Zuco V, De Cesare M, Zunino F, Simoes-Pires C, Nurisso A, Giannini G, Cuendet M, Dallavalle S. Cincinelli R, et al. Eur J Med Chem. 2016 Apr 13;112:99-105. doi: 10.1016/j.ejmech.2016.02.001. Epub 2016 Feb 3. Eur J Med Chem. 2016. PMID: 26890116 Free article.

3

Cell-based multi-substrate assay coupled to UHPLC-ESI-MS/MS for a quick identification of class-specific HDAC inhibitors.

Zwick V, Simões-Pires C, Cuendet M. Zwick V, et al. J Enzyme Inhib Med Chem. 2016;31(sup1):209-214. doi: 10.1080/14756366.2016.1180595. Epub 2016 May 5. J Enzyme Inhib Med Chem. 2016. PMID: 27149362

4

HDAC6 as a target for neurodegenerative diseases: what makes it different from the other HDACs?

Simões-Pires C, Zwick V, Nurisso A, Schenker E, Carrupt PA, Cuendet M. Simões-Pires C, et al. Mol Neurodegener. 2013 Jan 29;8:7. doi: 10.1186/1750-1326-8-7. Mol Neurodegener. 2013. PMID: 23356410 Free PMC article. Review.

5

Aurones as histone deacetylase inhibitors: identification of key features.

Zwick V, Chatzivasileiou AO, Deschamps N, Roussaki M, Simões-Pires CA, Nurisso A, Denis I, Blanquart C, Martinet N, Carrupt PA, Detsi A, Cuendet M. Zwick V, et al. Bioorg Med Chem Lett. 2014 Dec 1;24(23):5497-501. doi: 10.1016/j.bmcl.2014.10.019. Epub 2014 Oct 13. Bioorg Med Chem Lett. 2014. PMID: 25455492

6

Synthesis of a selective HDAC6 inhibitor active in neuroblasts.

Zwick V, Simões-Pires CA, Nurisso A, Petit C, Dos Santos Passos C, Randazzo GM, Martinet N, Bertrand P, Cuendet M. Zwick V, et al. Bioorg Med Chem Lett. 2016 Oct 15;26(20):4955-4959. doi: 10.1016/j.bmcl.2016.09.011. Epub 2016 Sep 7. Bioorg Med Chem Lett. 2016. PMID: 27650925

7

Novel histone deacetylase 6 (HDAC6) selective inhibitors: a patent evaluation (WO2014181137).

Simões-Pires CA, Bertrand P, Cuendet M. Simões-Pires CA, et al. Expert Opin Ther Pat. 2017 Mar;27(3):229-236. doi: 10.1080/13543776.2017.1282945. Epub 2017 Jan 31. Expert Opin Ther Pat. 2017. PMID: 28092474

8

How the flexibility of human histone deacetylases influences ligand binding: an overview.

Deschamps N, Simões-Pires CA, Carrupt PA, Nurisso A. Deschamps N, et al. Drug Discov Today. 2015 Jun;20(6):736-42. doi: 10.1016/j.drudis.2015.01.004. Epub 2015 Jan 15. Drug Discov Today. 2015. PMID: 25597521 Review.

9

A Rational Approach for the Identification of Non-Hydroxamate HDAC6-Selective Inhibitors.

Goracci L, Deschamps N, Randazzo GM, Petit C, Dos Santos Passos C, Carrupt PA, Simões-Pires C, Nurisso A. Goracci L, et al. Sci Rep. 2016 Jul 12;6:29086. doi: 10.1038/srep29086. Sci Rep. 2016. PMID: 27404291 Free PMC article.

10

UHPLC-MS-based HDAC Assay Applied to Bio-guided Microfractionation of Fungal Extracts.

Zwick V, Allard PM, Ory L, Simões-Pires CA, Marcourt L, Gindro K, Wolfender JL, Cuendet M. Zwick V, et al. Among authors: simoes pires ca. Phytochem Anal. 2017 Mar;28(2):93-100. doi: 10.1002/pca.2652. Epub 2016 Dec 5. Phytochem Anal. 2017. PMID: 27921344

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