Setola V - Search Results

1

Michael acceptor approach to the design of new salvinorin A-based high affinity ligands for the kappa-opioid receptor.

Polepally PR, Huben K, Vardy E, Setola V, Mosier PD, Roth BL, Zjawiony JK. Polepally PR, et al. Among authors: setola v. Eur J Med Chem. 2014 Oct 6;85:818-29. doi: 10.1016/j.ejmech.2014.07.077. Epub 2014 Aug 23. Eur J Med Chem. 2014. PMID: 25193297 Free PMC article.

2

Chemocentric informatics approach to drug discovery: identification and experimental validation of selective estrogen receptor modulators as ligands of 5-hydroxytryptamine-6 receptors and as potential cognition enhancers.

Hajjo R, Setola V, Roth BL, Tropsha A. Hajjo R, et al. Among authors: setola v. J Med Chem. 2012 Jun 28;55(12):5704-19. doi: 10.1021/jm2011657. Epub 2012 Jun 11. J Med Chem. 2012. PMID: 22537153 Free PMC article.

3

1-(1-Naphthyl)piperazine as a novel template for 5-HT6 serotonin receptor ligands.

Lee M, Rangisetty JB, Pullagurla MR, Dukat M, Setola V, Roth BL, Glennon RA. Lee M, et al. Among authors: setola v. Bioorg Med Chem Lett. 2005 Mar 15;15(6):1707-11. doi: 10.1016/j.bmcl.2005.01.031. Bioorg Med Chem Lett. 2005. PMID: 15745826

4

Interaction of chiral MS-245 analogs at h5-HT6 receptors.

Abate C, Kolanos R, Dukat M, Setola V, Roth BL, Glennon RA. Abate C, et al. Among authors: setola v. Bioorg Med Chem Lett. 2005 Aug 1;15(15):3510-3. doi: 10.1016/j.bmcl.2005.05.092. Bioorg Med Chem Lett. 2005. PMID: 15990303

5

N1-benzenesulfonylgramine and N1-benzenesulfonylskatole: novel 5-HT6 receptor ligand templates.

Pullagurla MR, Dukat M, Setola V, Roth B, Glennon RA. Pullagurla MR, et al. Among authors: setola v. Bioorg Med Chem Lett. 2003 Oct 6;13(19):3355-9. doi: 10.1016/s0960-894x(03)00612-7. Bioorg Med Chem Lett. 2003. PMID: 12951125

6

1,2,3,4-tetrahydrocarbazoles as 5-HT6 serotonin receptor ligands.

Chang-Fong J, Rangisetty JB, Dukat M, Setola V, Raffay T, Roth B, Glennon RA. Chang-Fong J, et al. Among authors: setola v. Bioorg Med Chem Lett. 2004 Apr 19;14(8):1961-4. doi: 10.1016/j.bmcl.2004.01.071. Bioorg Med Chem Lett. 2004. PMID: 15050637

7

Synthesis and evaluation of ligands for D2-like receptors: the role of common pharmacophoric groups.

Sikazwe DM, Nkansah NT, Altundas R, Zhu XY, Roth BL, Setola V, Ablordeppey SY. Sikazwe DM, et al. Among authors: setola v. Bioorg Med Chem. 2009 Feb 15;17(4):1716-23. doi: 10.1016/j.bmc.2008.12.054. Epub 2008 Dec 31. Bioorg Med Chem. 2009. PMID: 19155177 Free PMC article.

8

Improvement of pharmacological properties of irreversible thyroid receptor coactivator binding inhibitors.

Hwang JY, Arnold LA, Zhu F, Kosinski A, Mangano TJ, Setola V, Roth BL, Guy RK. Hwang JY, et al. Among authors: setola v. J Med Chem. 2009 Jul 9;52(13):3892-901. doi: 10.1021/jm9002704. J Med Chem. 2009. PMID: 19469546 Free PMC article.

9

N-Alkyl-octahydroisoquinolin-1-one-8-carboxamides: a Novel Class of Selective, Nonbasic, Nitrogen-Containing κ-Opioid Receptor Ligands.

Frankowski KJ, Ghosh P, Setola V, Tran TB, Roth BL, Aubé J. Frankowski KJ, et al. Among authors: setola v. ACS Med Chem Lett. 2010 Aug 12;1(5):189-193. doi: 10.1021/ml100040t. ACS Med Chem Lett. 2010. PMID: 20729985 Free PMC article.

10

Development, validation, and use of quantitative structure-activity relationship models of 5-hydroxytryptamine (2B) receptor ligands to identify novel receptor binders and putative valvulopathic compounds among common drugs.

Hajjo R, Grulke CM, Golbraikh A, Setola V, Huang XP, Roth BL, Tropsha A. Hajjo R, et al. Among authors: setola v. J Med Chem. 2010 Nov 11;53(21):7573-86. doi: 10.1021/jm100600y. J Med Chem. 2010. PMID: 20958049 Free PMC article.

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