Runyon SP - Search Results

1

Enhanced bioactivity of silybin B methylation products.

Sy-Cordero AA, Graf TN, Runyon SP, Wani MC, Kroll DJ, Agarwal R, Brantley SJ, Paine MF, Polyak SJ, Oberlies NH. Sy-Cordero AA, et al. Among authors: runyon sp. Bioorg Med Chem. 2013 Feb 1;21(3):742-7. doi: 10.1016/j.bmc.2012.11.035. Epub 2012 Dec 5. Bioorg Med Chem. 2013. PMID: 23260576 Free PMC article.

2

Monoamine transporter binding, locomotor activity, and drug discrimination properties of 3-(4-substituted-phenyl)tropane-2-carboxylic acid methyl ester isomers.

Carroll FI, Runyon SP, Abraham P, Navarro H, Kuhar MJ, Pollard GT, Howard JL. Carroll FI, et al. Among authors: runyon sp. J Med Chem. 2004 Dec 2;47(25):6401-9. doi: 10.1021/jm0401311. J Med Chem. 2004. PMID: 15566309

3

Synthesis, structural identification, and ligand binding of tropane ring analogs of paroxetine and an unexpected aza-bicyclo[3.2.2]nonane rearrangement product.

Runyon SP, Burgess JP, Abraham P, Keverline-Frantz KI, Flippen-Anderson J, Deschamps J, Lewin AH, Navarro HA, Boja JW, Kuhar MJ, Carroll FI. Runyon SP, et al. Bioorg Med Chem. 2005 Apr 1;13(7):2439-49. doi: 10.1016/j.bmc.2005.01.046. Bioorg Med Chem. 2005. PMID: 15755646

4

Identifying structural features on 1,1-diphenyl-hexahydro-oxazolo[3,4-a]pyrazin-3-ones critical for Neuropeptide S antagonist activity.

Zhang Y, Gilmour BP, Navarro HA, Runyon SP. Zhang Y, et al. Among authors: runyon sp. Bioorg Med Chem Lett. 2008 Jul 15;18(14):4064-7. doi: 10.1016/j.bmcl.2008.05.098. Epub 2008 Jun 12. Bioorg Med Chem Lett. 2008. PMID: 18555684 Free PMC article.

5

Analogues of (3R)-7-hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide (JDTic). Synthesis and in vitro and in vivo opioid receptor antagonist activity.

Runyon SP, Brieaddy LE, Mascarella SW, Thomas JB, Navarro HA, Howard JL, Pollard GT, Carroll FI. Runyon SP, et al. J Med Chem. 2010 Jul 22;53(14):5290-301. doi: 10.1021/jm1004978. J Med Chem. 2010. PMID: 20568781 Free PMC article.

6

Discovery of N-{4-[(3-hydroxyphenyl)-3-methylpiperazin-1-yl]methyl-2-methylpropyl}-4-phenoxybenzamide analogues as selective kappa opioid receptor antagonists.

Kormos CM, Jin C, Cueva JP, Runyon SP, Thomas JB, Brieaddy LE, Mascarella SW, Navarro HA, Gilmour BP, Carroll FI. Kormos CM, et al. Among authors: runyon sp. J Med Chem. 2013 Jun 13;56(11):4551-67. doi: 10.1021/jm400275h. Epub 2013 May 16. J Med Chem. 2013. PMID: 23651437 Free PMC article.

7

Effect of the 3- and 4-methyl groups on the opioid receptor properties of N-substituted trans-3,4-dimethyl-4-(3-hydroxyphenyl)piperidines.

Kormos CM, Cueva JP, Gichinga MG, Runyon SP, Thomas JB, Brieaddy LE, Mascarella SW, Gilmour BP, Navarro HA, Carroll FI. Kormos CM, et al. Among authors: runyon sp. J Med Chem. 2014 Apr 10;57(7):3140-7. doi: 10.1021/jm500184j. Epub 2014 Mar 26. J Med Chem. 2014. PMID: 24635568 Free PMC article.

8

Identifying structural determinants of potency for analogs of apelin-13: integration of C-terminal truncation with structure-activity.

Zhang Y, Maitra R, Harris DL, Dhungana S, Snyder R, Runyon SP. Zhang Y, et al. Among authors: runyon sp. Bioorg Med Chem. 2014 Jun 1;22(11):2992-7. doi: 10.1016/j.bmc.2014.04.001. Epub 2014 Apr 13. Bioorg Med Chem. 2014. PMID: 24755525

9

Identification of 1-({[1-(4-fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)cyclohexane carboxylic acid as a selective nonpeptide neurotensin receptor type 2 compound.

Thomas JB, Giddings AM, Wiethe RW, Olepu S, Warner KR, Sarret P, Gendron L, Longpre JM, Zhang Y, Runyon SP, Gilmour BP. Thomas JB, et al. Among authors: runyon sp. J Med Chem. 2014 Jun 26;57(12):5318-32. doi: 10.1021/jm5003843. Epub 2014 Jun 5. J Med Chem. 2014. PMID: 24856674 Free PMC article.

10

Identification of neuropeptide S antagonists: structure-activity relationship studies, X-ray crystallography, and in vivo evaluation.

Hassler C, Zhang Y, Gilmour B, Graf T, Fennell T, Snyder R, Deschamps JR, Reinscheid RK, Garau C, Runyon SP. Hassler C, et al. Among authors: runyon sp. ACS Chem Neurosci. 2014 Aug 20;5(8):731-44. doi: 10.1021/cn500113c. Epub 2014 Jul 11. ACS Chem Neurosci. 2014. PMID: 24964000 Free PMC article.

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