Steelman G - Search Results

1

Synthesis and SAR of aminothiazole fused benzazepines as selective dopamine D2 partial agonists.

Urbanek RA, Xiong H, Wu Y, Blackwell W, Steelman G, Rosamond J, Wesolowski SS, Campbell JB, Zhang M, Brockel B, Widzowski DV. Urbanek RA, et al. Among authors: steelman g. Bioorg Med Chem Lett. 2013 Jan 15;23(2):543-7. doi: 10.1016/j.bmcl.2012.11.023. Epub 2012 Nov 28. Bioorg Med Chem Lett. 2013. PMID: 23237836

2

Synthesis of 7-chloro-2,3-dihydro-2-[1-(pyridinyl)alkyl]-pyridazino[4,5-b]quinoline-1,4,10(5H)-triones as NMDA glycine-site antagonists.

Brown DG, Urbanek RA, Bare TM, McLaren FM, Horchler CL, Murphy M, Steelman GB, Empfield JR, Forst JM, Herzog KJ, Xiao W, Dyroff MC, Lee CM, Trivedi S, Neilson KL, Keith RA. Brown DG, et al. Among authors: steelman gb. Bioorg Med Chem Lett. 2003 Oct 20;13(20):3553-6. doi: 10.1016/s0960-894x(03)00750-9. Bioorg Med Chem Lett. 2003. PMID: 14505669

3

Pyridazinoquinolinetriones as NMDA glycine-site antagonists with oral antinociceptive activity in a model of neuropathic pain.

Bare TM, Brown DG, Horchler CL, Murphy M, Urbanek RA, Alford V, Barlaam C, Dyroff MC, Empfield JB, Forst JM, Herzog KJ, Keith RA, Kirschner AS, Lee CM, Lewis J, McLaren FM, Neilson KL, Steelman GB, Trivedi S, Vacek EP, Xiao W. Bare TM, et al. Among authors: steelman gb. J Med Chem. 2007 Jun 28;50(13):3113-31. doi: 10.1021/jm060212s. Epub 2007 Jun 2. J Med Chem. 2007. PMID: 17542571

4

Azepines and piperidines with dual norepinephrine dopamine uptake inhibition and antidepressant activity.

Brown DG, Bernstein PR, Wu Y, Urbanek RA, Becker CW, Throner SR, Dembofsky BT, Steelman GB, Lazor LA, Scott CW, Wood MW, Wesolowski SS, Nugiel DA, Koch S, Yu J, Pivonka DE, Li S, Thompson C, Zacco A, Elmore CS, Schroeder P, Liu J, Hurley CA, Ward S, Hunt HJ, Williams K, McLaughlin J, Hoesch V, Sydserff S, Maier D, Aharony D. Brown DG, et al. Among authors: steelman gb. ACS Med Chem Lett. 2012 Nov 12;4(1):46-51. doi: 10.1021/ml300262e. eCollection 2013 Jan 10. ACS Med Chem Lett. 2012. PMID: 24900562 Free PMC article.

5

Potent reversible inhibitors of the protein tyrosine phosphatase CD45.

Urbanek RA, Suchard SJ, Steelman GB, Knappenberger KS, Sygowski LA, Veale CA, Chapdelaine MJ. Urbanek RA, et al. Among authors: steelman gb. J Med Chem. 2001 May 24;44(11):1777-93. doi: 10.1021/jm000447i. J Med Chem. 2001. PMID: 11356112

6

Bicyclo((aryl)methyl)benzamides as inhibitors of GlyT1.

Varnes JG, Xiong H, Forst JM, Holmquist CR, Ernst GE, Frietze W, Dembofsky B, Andisik DW, Palmer WE, Hinkley L, Steelman GB, Wilkins DE, Tian G, Jonak G, Potts WM, Wang X, Brugel TA, Alhambra C, Wood MW, Veale CA, Albert JS. Varnes JG, et al. Among authors: steelman gb. Bioorg Med Chem Lett. 2018 Apr 1;28(6):1043-1049. doi: 10.1016/j.bmcl.2018.02.029. Epub 2018 Feb 14. Bioorg Med Chem Lett. 2018. PMID: 29486970

7

The discovery of non-basic atrial natriuretic peptide clearance receptor antagonists. Part 1.

Veale CA, Alford VC, Aharony D, Banville DL, Bialecki RA, Brown FJ, Damewood JR Jr, Dantzman CL, Edwards PD, Jacobs RT, Mauger RC, Murphy MM, Palmer W, Pine KK, Rumsey WL, Garcia-Davenport LE, Shaw A, Steelman GB, Surian JM, Vacek EP. Veale CA, et al. Among authors: steelman gb. Bioorg Med Chem Lett. 2000 Sep 4;10(17):1949-52. doi: 10.1016/s0960-894x(00)00387-5. Bioorg Med Chem Lett. 2000. PMID: 10987424

8

Nonpeptidic inhibitors of human leukocyte elastase. 5. Design, synthesis, and X-ray crystallography of a series of orally active 5-aminopyrimidin-6-one-containing trifluoromethyl ketones.

Veale CA, Bernstein PR, Bryant C, Ceccarelli C, Damewood JR Jr, Earley R, Feeney SW, Gomes B, Kosmider BJ, Steelman GB, et al. Veale CA, et al. Among authors: steelman gb. J Med Chem. 1995 Jan 6;38(1):98-108. doi: 10.1021/jm00001a015. J Med Chem. 1995. PMID: 7837246

9

Nonpeptidic inhibitors of human leukocyte elastase. 2. Design, synthesis, and in vitro activity of a series of 3-amino-6-arylopyridin-2-one trifluoromethyl ketones.

Damewood JR Jr, Edwards PD, Feeney S, Gomes BC, Steelman GB, Tuthill PA, Williams JC, Warner P, Woolson SA, Wolanin DJ, et al. Damewood JR Jr, et al. Among authors: steelman gb. J Med Chem. 1994 Sep 30;37(20):3303-12. doi: 10.1021/jm00046a015. J Med Chem. 1994. PMID: 7932558

10

Non-peptidic inhibitors of human leukocyte elastase. 4. Design, synthesis, and in vitro and in vivo activity of a series of beta-carbolinone-containing trifluoromethyl ketones.

Veale CA, Damewood JR Jr, Steelman GB, Bryant C, Gomes B, Williams J. Veale CA, et al. Among authors: steelman gb. J Med Chem. 1995 Jan 6;38(1):86-97. doi: 10.1021/jm00001a014. J Med Chem. 1995. PMID: 7837244

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