Augustyns K - Search Results

1

Synthesis, evaluation and structure-activity relationships of triazine dimers as novel antiviral agents.

Venkatraj M, Ariën KK, Heeres J, Joossens J, Messagie J, Michiels J, Van der Veken P, Vanham G, Lewi PJ, Augustyns K. Venkatraj M, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2012 Dec 1;22(23):7174-8. doi: 10.1016/j.bmcl.2012.09.066. Epub 2012 Sep 27. Bioorg Med Chem Lett. 2012. PMID: 23084903

2

Synthesis and anti-HIV evaluation of 2',3'-dideoxyribo-5-chloropyrimidine analogues: reduced toxicity of 5-chlorinated 2',3'-dideoxynucleosides.

Van Aerschot A, Everaert D, Balzarini J, Augustyns K, Jie L, Janssen G, Peeters O, Blaton N, De Ranter C, De Clercq E, et al. Van Aerschot A, et al. Among authors: augustyns k. J Med Chem. 1990 Jun;33(6):1833-9. doi: 10.1021/jm00168a046. J Med Chem. 1990. PMID: 2342078

3

Structure-activity relationship of diaryl phosphonate esters as potent irreversible dipeptidyl peptidase IV inhibitors.

Belyaev A, Zhang X, Augustyns K, Lambeir AM, De Meester I, Vedernikova I, Scharpé S, Haemers A. Belyaev A, et al. Among authors: augustyns k. J Med Chem. 1999 Mar 25;42(6):1041-52. doi: 10.1021/jm981033g. J Med Chem. 1999. PMID: 10090787

4

Synthesis and evaluation of caffeic acid amides as antioxidants.

Rajan P, Vedernikova I, Cos P, Berghe DV, Augustyns K, Haemers A. Rajan P, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2001 Jan 22;11(2):215-7. doi: 10.1016/s0960-894x(00)00630-2. Bioorg Med Chem Lett. 2001. PMID: 11206462

5

Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 1: Substitution of the glycine carboxylic acid group.

Amssoms K, Oza SL, Ravaschino E, Yamani A, Lambeir A, Rajan P, Bal G, Rodriguez J, Fairlamb AH, Augustyns K, Haemers A. Amssoms K, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2002 Sep 16;12(18):2553-6. doi: 10.1016/s0960-894x(02)00489-4. Bioorg Med Chem Lett. 2002. PMID: 12182858

6

Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 2: substitution of the glycine part.

Amssoms K, Oza SL, Augustyns K, Yamani A, Lambeir AM, Bal G, Van der Veken P, Fairlamb AH, Haemers A. Amssoms K, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2002 Oct 7;12(19):2703-5. doi: 10.1016/s0960-894x(02)00538-3. Bioorg Med Chem Lett. 2002. PMID: 12217358

7

Development of potent and selective dipeptidyl peptidase II inhibitors.

Senten K, Van der Veken P, Bal G, De Meester I, Lambeir AM, Scharpé S, Bauvois B, Haemers A, Augustyns K. Senten K, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2002 Oct 21;12(20):2825-8. doi: 10.1016/s0960-894x(02)00603-0. Bioorg Med Chem Lett. 2002. PMID: 12270155

8

Rapid parallel synthesis of dipeptide diphenyl phosphonate esters as inhibitors of dipeptidyl peptidases.

Senten K, Daniëls L, Van der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: augustyns k. J Comb Chem. 2003 May-Jun;5(3):336-44. doi: 10.1021/cc020096o. J Comb Chem. 2003. PMID: 12739951

9

Design, synthesis, and SAR of potent and selective dipeptide-derived inhibitors for dipeptidyl peptidases.

Senten K, Van der Veken P, De Meester I, Lambeir AM, Scharpé S, Haemers A, Augustyns K. Senten K, et al. Among authors: augustyns k. J Med Chem. 2003 Nov 6;46(23):5005-14. doi: 10.1021/jm0308803. J Med Chem. 2003. PMID: 14584950

10

Prolylisoxazoles: potent inhibitors of prolyloligopeptidase with antitrypanosomal activity.

Bal G, Van der Veken P, Antonov D, Lambeir AM, Grellier P, Croft SL, Augustyns K, Haemers A. Bal G, et al. Among authors: augustyns k. Bioorg Med Chem Lett. 2003 Sep 1;13(17):2875-8. doi: 10.1016/s0960-894x(03)00579-1. Bioorg Med Chem Lett. 2003. PMID: 14611847

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