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Discovery of N-benzyl-2-[(4S)-4-(1H-indol-3-ylmethyl)-5-oxo-1-phenyl-4,5-dihydro-6H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-6-yl]-N-isopropylacetamide, an orally active, gut-selective CCK1 receptor agonist for the potential treatment of obesity.
Bioorg Med Chem Lett. 2010 Nov 15;20(22):6797-801. doi: 10.1016/j.bmcl.2010.08.115. Epub 2010 Sep 28.
Bioorg Med Chem Lett. 2010.
PMID: 20851601
Discovery of potent, nonsteroidal, and highly selective glucocorticoid receptor antagonists.
Morgan BP, Swick AG, Hargrove DM, LaFlamme JA, Moynihan MS, Carroll RS, Martin KA, Lee E, Decosta D, Bordner J.
Morgan BP, et al. Among authors: laflamme ja.
J Med Chem. 2002 Jun 6;45(12):2417-24. doi: 10.1021/jm0105530.
J Med Chem. 2002.
PMID: 12036351
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Structure-activity relationships in a series of NPY Y5 antagonists: 3-amido-9-ethylcarbazoles, core-modified analogues and amide isosteres.
Hammond M, Elliott RL, Gillaspy ML, Hager DC, Hank RF, LaFlamme JA, Oliver RM, DaSilva-Jardine PA, Stevenson RW, Mack CM, Cassella JV.
Hammond M, et al. Among authors: laflamme ja.
Bioorg Med Chem Lett. 2003 Jun 16;13(12):1989-92. doi: 10.1016/s0960-894x(03)00329-9.
Bioorg Med Chem Lett. 2003.
PMID: 12781180
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Structure-activity relationship studies on 2-heteroaryl-4-arylimidazoles NPY5 receptor antagonists.
Elliott RL, Oliver RM, LaFlamme JA, Gillaspy ML, Hammond M, Hank RF, Maurer TS, Baker DL, DaSilva-Jardine PA, Stevenson RW, Mack CM, Cassella JV.
Elliott RL, et al. Among authors: laflamme ja.
Bioorg Med Chem Lett. 2003 Oct 20;13(20):3593-6. doi: 10.1016/s0960-894x(03)00747-9.
Bioorg Med Chem Lett. 2003.
PMID: 14505677
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