Casara PJ - Search Results

1

Blockade of alpha v beta3 and alpha v beta5 integrins by RGD mimetics induces anoikis and not integrin-mediated death in human endothelial cells.

Maubant S, Saint-Dizier D, Boutillon M, Perron-Sierra F, Casara PJ, Hickman JA, Tucker GC, Van Obberghen-Schilling E. Maubant S, et al. Among authors: casara pj. Blood. 2006 Nov 1;108(9):3035-44. doi: 10.1182/blood-2006-05-023580. Epub 2006 Jul 11. Blood. 2006. PMID: 16835373 Free article.

2

Substituted benzocyloheptenes as potent and selective alpha(v) integrin antagonists.

Perron-Sierra F, Saint Dizier D, Bertrand M, Genton A, Tucker GC, Casara P. Perron-Sierra F, et al. Bioorg Med Chem Lett. 2002 Nov 18;12(22):3291-6. doi: 10.1016/s0960-894x(02)00696-0. Bioorg Med Chem Lett. 2002. PMID: 12392735

3

Decrease in survival threshold of quiescent colon carcinoma cells in the presence of a small molecule integrin antagonist.

Burbridge MF, Venot V, Casara PJ, Perron-Sierra F, Hickman JA, Tucker GC. Burbridge MF, et al. Among authors: casara pj. Mol Pharmacol. 2003 Jun;63(6):1281-8. doi: 10.1124/mol.63.6.1281. Mol Pharmacol. 2003. PMID: 12761337

4

Bax activation by engagement with, then release from, the BH3 binding site of Bcl-xL.

Gautier F, Guillemin Y, Cartron PF, Gallenne T, Cauquil N, Le Diguarher T, Casara P, Vallette FM, Manon S, Hickman JA, Geneste O, Juin P. Gautier F, et al. Mol Cell Biol. 2011 Feb;31(4):832-44. doi: 10.1128/MCB.00161-10. Epub 2010 Dec 20. Mol Cell Biol. 2011. PMID: 21173168 Free PMC article.

5

Parallel liquid synthesis of N,N'-Disubstituted 3-amino azepin-2-ones as potent and specific farnesyl transferase inhibitors.

Le Diguarher T, Ortuno JC, Dorey G, Shanks D, Guilbaud N, Pierré A, Fauchère JL, Hickman JA, Tucker GC, Casara PJ. Le Diguarher T, et al. Among authors: casara pj. Bioorg Med Chem. 2003 Jul 17;11(14):3193-204. doi: 10.1016/s0968-0896(03)00218-9. Bioorg Med Chem. 2003. PMID: 12818682

6

Synthesis of N,N'-disubstituted 3-aminobenzo[c] and [d]azepin-2-ones as potent and specific farnesyl transferase inhibitors.

Le Diguarher T, Ortuno JC, Shanks D, Guilbaud N, Pierré A, Raimbaud E, Fauchère JL, Hickman JA, Tucker GC, Casara PJ. Le Diguarher T, et al. Among authors: casara pj. Bioorg Med Chem Lett. 2004 Feb 9;14(3):767-71. doi: 10.1016/j.bmcl.2003.11.013. Bioorg Med Chem Lett. 2004. PMID: 14741286

7

S55746 is a novel orally active BCL-2 selective and potent inhibitor that impairs hematological tumor growth.

Casara P, Davidson J, Claperon A, Le Toumelin-Braizat G, Vogler M, Bruno A, Chanrion M, Lysiak-Auvity G, Le Diguarher T, Starck JB, Chen I, Whitehead N, Graham C, Matassova N, Dokurno P, Pedder C, Wang Y, Qiu S, Girard AM, Schneider E, Gravé F, Studeny A, Guasconi G, Rocchetti F, Maïga S, Henlin JM, Colland F, Kraus-Berthier L, Le Gouill S, Dyer MJS, Hubbard R, Wood M, Amiot M, Cohen GM, Hickman JA, Morris E, Murray J, Geneste O. Casara P, et al. Oncotarget. 2018 Apr 13;9(28):20075-20088. doi: 10.18632/oncotarget.24744. eCollection 2018 Apr 13. Oncotarget. 2018. PMID: 29732004 Free PMC article.

8

General synthesis of alpha-substituted 3-bisaryloxy propionic acid derivatives as specific MMP inhibitors.

Chollet AM, Le Diguarher T, Murray L, Bertrand M, Tucker GC, Sabatini M, Pierré A, Atassi G, Bonnet J, Casara P. Chollet AM, et al. Bioorg Med Chem Lett. 2001 Feb 12;11(3):295-9. doi: 10.1016/s0960-894x(00)00646-6. Bioorg Med Chem Lett. 2001. PMID: 11212095

9

Stereospecific synthesis of 5-substituted 2-bisarylthiocyclopentane carboxylic acids as specific matrix metalloproteinase inhibitors.

Le Diguarher T, Chollet AM, Bertrand M, Hennig P, Raimbaud E, Sabatini M, Guilbaud N, Pierré A, Tucker GC, Casara P. Le Diguarher T, et al. J Med Chem. 2003 Aug 28;46(18):3840-52. doi: 10.1021/jm0307638. J Med Chem. 2003. PMID: 12930146

10

Synthesis of Cis-fused pyran indolocarbazole derivatives that inhibit FLT3 kinase and the DNA damage kinase, checkpoint kinase 1.

Perron-Sierra FM, Kucharkzyk N, Boucley C, Guyard-Daumas C, Sciberras S, Fouache C, Plantier S, Studeny A, Bossard C, Casara PJ, Golsteyn RM. Perron-Sierra FM, et al. Among authors: casara pj. Anticancer Agents Med Chem. 2012 Mar;12(3):194-201. doi: 10.2174/187152012800228823. Anticancer Agents Med Chem. 2012. PMID: 22044003

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