Vinader VM - Search Results

1

Dissociated nonsteroidal glucocorticoid receptor modulators; discovery of the agonist trigger in a tetrahydronaphthalene-benzoxazine series.

Barker M, Clackers M, Copley R, Demaine DA, Humphreys D, Inglis GG, Johnston MJ, Jones HT, Haase MV, House D, Loiseau R, Nisbet L, Pacquet F, Skone PA, Shanahan SE, Tape D, Vinader VM, Washington M, Uings I, Upton R, McLay IM, Macdonald SJ. Barker M, et al. Among authors: vinader vm. J Med Chem. 2006 Jul 13;49(14):4216-31. doi: 10.1021/jm060302x. J Med Chem. 2006. PMID: 16821781

2

Design and synthesis of new nonsteroidal glucocorticoid modulators through application of an "agreement docking" method.

Barker M, Clackers M, Demaine DA, Humphreys D, Johnston MJ, Jones HT, Pacquet F, Pritchard JM, Salter M, Shanahan SE, Skone PA, Vinader VM, Uings I, McLay IM, Macdonald SJ. Barker M, et al. Among authors: vinader vm. J Med Chem. 2005 Jul 14;48(14):4507-10. doi: 10.1021/jm050345y. J Med Chem. 2005. PMID: 15999989

3

Oxazolidinones as novel human CCR8 antagonists.

Jin J, Wang Y, Wang F, Kerns JK, Vinader VM, Hancock AP, Lindon MJ, Stevenson GI, Morrow DM, Rao P, Nguyen C, Barrett VJ, Browning C, Hartmann G, Andrew DP, Sarau HM, Foley JJ, Jurewicz AJ, Fornwald JA, Harker AJ, Moore ML, Rivero RA, Belmonte KE, Connor HE. Jin J, et al. Among authors: vinader vm. Bioorg Med Chem Lett. 2007 Mar 15;17(6):1722-5. doi: 10.1016/j.bmcl.2006.12.076. Epub 2006 Dec 24. Bioorg Med Chem Lett. 2007. PMID: 17267215

4

1 alpha,25-dihydroxyvitamin D3 analogs featuring aromatic and heteroaromatic rings: design, synthesis, and preliminary biological testing.

Posner GH, Li Z, White MC, Vinader V, Takeuchi K, Guggino SE, Dolan P, Kensler TW. Posner GH, et al. J Med Chem. 1995 Oct 27;38(22):4529-37. doi: 10.1021/jm00022a019. J Med Chem. 1995. PMID: 7473581

5

Synthesis and biological evaluation of colchicine B-ring analogues tethered with halogenated benzyl moieties.

Cosentino L, Redondo-Horcajo M, Zhao Y, Santos AR, Chowdury KF, Vinader V, Abdallah QM, Abdel-Rahman H, Fournier-Dit-Chabert J, Shnyder SD, Loadman PM, Fang WS, Díaz JF, Barasoain I, Burns PA, Pors K. Cosentino L, et al. J Med Chem. 2012 Dec 27;55(24):11062-6. doi: 10.1021/jm301151t. Epub 2012 Dec 7. J Med Chem. 2012. PMID: 23176628

6

Molybdenum(IV) Complexes as Efficient, Lewis Acidic Catalysts for Allylic Substitution. Formation of C-C and C-N Bonds.

Malkov AV, Spoor P, Vinader V, Kočovský P. Malkov AV, et al. J Org Chem. 1999 Jul 9;64(14):5308-5311. doi: 10.1021/jo990372u. J Org Chem. 1999. PMID: 34237862 No abstract available.

7

Discovery and computer aided potency optimization of a novel class of small molecule CXCR4 antagonists.

Vinader V, Ahmet DS, Ahmed MS, Patterson LH, Afarinkia K. Vinader V, et al. PLoS One. 2013 Oct 18;8(10):e78744. doi: 10.1371/journal.pone.0078744. eCollection 2013. PLoS One. 2013. PMID: 24205302 Free PMC article.

8

Synthesis and biological evaluation of colchicine C-ring analogues tethered with aliphatic linkers suitable for prodrug derivatisation.

Fournier-Dit-Chabert J, Vinader V, Santos AR, Redondo-Horcajo M, Dreneau A, Basak R, Cosentino L, Marston G, Abdel-Rahman H, Loadman PM, Shnyder SD, Díaz JF, Barasoain I, Falconer RA, Pors K. Fournier-Dit-Chabert J, et al. Bioorg Med Chem Lett. 2012 Dec 15;22(24):7693-6. doi: 10.1016/j.bmcl.2012.09.104. Epub 2012 Oct 10. Bioorg Med Chem Lett. 2012. PMID: 23103097

9

Asymmetric allylic substitution catalyzed by C1-symmetrical complexes of molybdenum: structural requirements of the ligand and the stereochemical course of the reaction.

Malkov AV, Gouriou L, Lloyd-Jones GC, Starý I, Langer V, Spoor P, Vinader V, Kocovský P. Malkov AV, et al. Chemistry. 2006 Sep 6;12(26):6910-29. doi: 10.1002/chem.200501574. Chemistry. 2006. PMID: 16807930

10

Synthesis of a pseudo-disaccharide library and its application to the characterisation of the heparanase catalytic site.

Vinader V, Haji-Abdullahi MH, Patterson LH, Afarinkia K. Vinader V, et al. PLoS One. 2013 Nov 18;8(11):e82111. doi: 10.1371/journal.pone.0082111. eCollection 2013. PLoS One. 2013. PMID: 24260588 Free PMC article.

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