Szardenings AK - Search Results

1

Synthesis and structure-activity relationship of N-alkyl Gly-boro-Pro inhibitors of DPP4, FAP, and DPP7.

Hu Y, Ma L, Wu M, Wong MS, Li B, Corral S, Yu Z, Nomanbhoy T, Alemayehu S, Fuller SR, Rosenblum JS, Rozenkrants N, Minimo LC, Ripka WC, Szardenings AK, Kozarich JW, Shreder KR. Hu Y, et al. Among authors: szardenings ak. Bioorg Med Chem Lett. 2005 Oct 1;15(19):4239-42. doi: 10.1016/j.bmcl.2005.06.075. Bioorg Med Chem Lett. 2005. PMID: 16085416

2

Synthesis and structure-activity relationship of 4-quinolone-3-carboxylic acid based inhibitors of glycogen synthase kinase-3β.

Cociorva OM, Li B, Nomanbhoy T, Li Q, Nakamura A, Nakamura K, Nomura M, Okada K, Seto S, Yumoto K, Liyanage M, Zhang MC, Aban A, Leen B, Szardenings AK, Rosenblum JS, Kozarich JW, Kohno Y, Shreder KR. Cociorva OM, et al. Among authors: szardenings ak. Bioorg Med Chem Lett. 2011 Oct 1;21(19):5948-51. doi: 10.1016/j.bmcl.2011.07.073. Epub 2011 Aug 5. Bioorg Med Chem Lett. 2011. PMID: 21873061

3

6-Position optimization of tricyclic 4-quinolone-based inhibitors of glycogen synthase kinase-3β: discovery of nitrile derivatives with picomolar potency.

Li B, Cociorva OM, Nomanbhoy T, Li Q, Nakamura K, Nomura M, Okada K, Yumoto K, Liyanage M, Zhang MC, Aban A, Szardenings AK, Kozarich JW, Kohno Y, Shreder KR. Li B, et al. Among authors: szardenings ak. Bioorg Med Chem Lett. 2012 Jan 15;22(2):1005-8. doi: 10.1016/j.bmcl.2011.12.006. Epub 2011 Dec 8. Bioorg Med Chem Lett. 2012. PMID: 22202172

4

Design and synthesis of AX4697, a bisindolylmaleimide exo-affinity probe that labels protein kinase C alpha and beta.

Liu Y, Wu J, Weissig H, Betancort JM, Gai WZ, Leventhal PS, Patricelli MP, Samii B, Szardenings AK, Shreder KR, Kozarich JW. Liu Y, et al. Among authors: szardenings ak. Bioorg Med Chem Lett. 2008 Nov 15;18(22):5955-8. doi: 10.1016/j.bmcl.2008.08.045. Epub 2008 Aug 19. Bioorg Med Chem Lett. 2008. PMID: 18774710

5

Synthesis and activity of a potent, specific azabicyclo[3.3.0]-octane-based DPP II inhibitor.

Danilova O, Li B, Szardenings AK, Huber BT, Rosenblum JS. Danilova O, et al. Among authors: szardenings ak. Bioorg Med Chem Lett. 2007 Jan 15;17(2):507-10. doi: 10.1016/j.bmcl.2006.10.012. Epub 2006 Oct 10. Bioorg Med Chem Lett. 2007. PMID: 17055271 Free PMC article.

6

Functional interrogation of the kinome using nucleotide acyl phosphates.

Patricelli MP, Szardenings AK, Liyanage M, Nomanbhoy TK, Wu M, Weissig H, Aban A, Chun D, Tanner S, Kozarich JW. Patricelli MP, et al. Among authors: szardenings ak. Biochemistry. 2007 Jan 16;46(2):350-8. doi: 10.1021/bi062142x. Biochemistry. 2007. PMID: 17209545

7

2,5-Diketopiperazines as potent and selective oxytocin antagonists 1: Identification, stereochemistry and initial SAR.

Wyatt PG, Allen MJ, Borthwick AD, Davies DE, Exall AM, Hatley RJ, Irving WR, Livermore DG, Miller ND, Nerozzi F, Sollis SL, Szardenings AK. Wyatt PG, et al. Among authors: szardenings ak. Bioorg Med Chem Lett. 2005 May 16;15(10):2579-82. doi: 10.1016/j.bmcl.2005.03.045. Bioorg Med Chem Lett. 2005. PMID: 15863320

8

Alpha,alpha-difluoro-beta-ketophosphonates as potent inhibitors of protein tyrosine phosphatase 1B.

Li X, Bhandari A, Holmes CP, Szardenings AK. Li X, et al. Among authors: szardenings ak. Bioorg Med Chem Lett. 2004 Aug 16;14(16):4301-6. doi: 10.1016/j.bmcl.2004.05.082. Bioorg Med Chem Lett. 2004. PMID: 15261291

9

Identification of highly selective inhibitors of collagenase-1 from combinatorial libraries of diketopiperazines.

Szardenings AK, Antonenko V, Campbell DA, DeFrancisco N, Ida S, Shi L, Sharkov N, Tien D, Wang Y, Navre M. Szardenings AK, et al. J Med Chem. 1999 Apr 22;42(8):1348-57. doi: 10.1021/jm980475p. J Med Chem. 1999. PMID: 10212120

10

Rational design and combinatorial evaluation of enzyme inhibitor scaffolds: identification of novel inhibitors of matrix metalloproteinases.

Szardenings AK, Harris D, Lam S, Shi L, Tien D, Wang Y, Patel DV, Navre M, Campbell DA. Szardenings AK, et al. J Med Chem. 1998 Jun 18;41(13):2194-200. doi: 10.1021/jm980133j. J Med Chem. 1998. PMID: 9632351

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