The target of ezetimibe is Niemann-Pick C1-Like 1 (NPC1L1).
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Proc Natl Acad Sci U S A. 2005 Jun 7;102(23):8132-7. doi: 10.1073/pnas.0500269102. Epub 2005 May 31.
Proc Natl Acad Sci U S A. 2005.
PMID: 15928087
Free PMC article.