Numazawa M - Search Results

1

Role of hydrophilic interaction in binding of hydroxylated 3-deoxy C(19) steroids to the active site of aromatase.

Numazawa M, Yamada K, Nitta S, Sasaki C, Kidokoro K. Numazawa M, et al. J Med Chem. 2001 Nov 22;44(24):4277-83. doi: 10.1021/jm010282t. J Med Chem. 2001. PMID: 11708928

2

Synthesis and biochemical properties of 6-bromoandrostenedione derivatives with a 2,2-dimethyl or 2-methyl group as aromatase inhibitors.

Numazawa M, Handa W, Yamada K. Numazawa M, et al. Biol Pharm Bull. 2004 Nov;27(11):1878-82. doi: 10.1248/bpb.27.1878. Biol Pharm Bull. 2004. PMID: 15516742 Free article.

3

Synthesis of 19-oxygenated derivatives of the competitive inhibitor of aromatase, 5-androstene-4,17-dione.

Numazawa M, Yamada K. Numazawa M, et al. Steroids. 1999 May;64(5):320-7. doi: 10.1016/s0039-128x(98)00113-5. Steroids. 1999. PMID: 10406481

4

19-oxygenated derivatives of androst-4-ene-6,17-dione and androst-5-ene-4,17-dione as catalytic probes for the active site of aromatase.

Numazawa M, Yamada K, Kidokoro K. Numazawa M, et al. Biol Pharm Bull. 1999 Oct;22(10):1134-6. doi: 10.1248/bpb.22.1134. Biol Pharm Bull. 1999. PMID: 10549872 Free article.

5

Studies of the time-dependent inactivation of aromatase by 4beta,5beta-epoxy-6-one and 5beta,6beta-epoxy-4-one steroids under various conditions.

Numazawa M, Yamada K. Numazawa M, et al. Biol Pharm Bull. 1999 Nov;22(11):1207-11. doi: 10.1248/bpb.22.1207. Biol Pharm Bull. 1999. PMID: 10598029 Free article.

6

19-Oxygenation of C19-steroids with an A, B-ring enone structure, competitive inhibitors of estrogen biosynthesis, with human placental aromatase.

Numazawa M, Yamada K, Nagaoka M. Numazawa M, et al. Biol Pharm Bull. 2001 Apr;24(4):332-5. doi: 10.1248/bpb.24.332. Biol Pharm Bull. 2001. PMID: 11305590 Free article.

7

Probing the active site of aromatase with 2-methyl-substituted androstenedione analogs.

Numazawa M, Watari Y, Yamada K, Umemura N, Handa W. Numazawa M, et al. Steroids. 2003 Aug;68(6):503-13. doi: 10.1016/s0039-128x(03)00089-8. Steroids. 2003. PMID: 12906935

8

Structure-activity relationships of 3-deoxy androgens as aromatase inhibitors. Synthesis and biochemical studies of 4-substituted 4-ene and 5-ene steroids.

Nagaoka M, Watari Y, Yajima H, Tsukioka K, Muroi Y, Yamada K, Numazawa M. Nagaoka M, et al. Among authors: numazawa m. Steroids. 2003 Aug;68(6):533-42. doi: 10.1016/s0039-128x(03)00085-0. Steroids. 2003. PMID: 12906938

9

Improved synthesis and molecular modeling of 4beta,19-dihydroxyandrost-5-en-17-one, an excellent inhibitor of aromatase.

Numazawa M, Yamada K, Watari Y, Ando M. Numazawa M, et al. Chem Pharm Bull (Tokyo). 2002 May;50(5):703-5. doi: 10.1248/cpb.50.703. Chem Pharm Bull (Tokyo). 2002. PMID: 12036037 Free article.

10

Synthesis of androst-5-en-7-ones and androsta-3,5-dien-7-ones and their related 7-deoxy analogs as conformational and catalytic probes for the active site of aromatase.

Numazawa M, Mutsumi A, Tachibana M, Hoshi K. Numazawa M, et al. J Med Chem. 1994 Jul 8;37(14):2198-205. doi: 10.1021/jm00040a012. J Med Chem. 1994. PMID: 8035427

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