Arachidonic acid activates a proton current in the rat glutamate transporter EAAT4

J Biol Chem. 1998 Jul 10;273(28):17315-7. doi: 10.1074/jbc.273.28.17315.

Abstract

The excitatory amino acid transporter EAAT4 is expressed predominantly in Purkinje neurons in the rat cerebellum (1-3), and it participates in postsynaptic reuptake of glutamate released at the climbing fiber synapse (4). Transporter-mediated currents in Purkinje neurons are increased more than 3-fold by arachidonic acid, a second messenger that is liberated following depolarization-induced Ca2+ activation of phospholipase A2 (5). In this study we demonstrate that application of arachidonic acid to oocytes expressing rat EAAT4 increased glutamate-induced currents to a similar extent. However, arachidonic acid did not cause an increase in the rate of glutamate transport or in the chloride current associated with glutamate transport but rather activated a proton-selective conductance. These data reveal a novel action of arachidonate on a glutamate transporter and suggest a mechanism by which synaptic activity may decrease intracellular pH in neurons where this transporter is localized.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Transport System X-AG*
  • Animals
  • Arachidonic Acid / pharmacology*
  • Excitatory Amino Acid Transporter 4
  • Glutamate Plasma Membrane Transport Proteins
  • Protons*
  • Purkinje Cells / drug effects*
  • Purkinje Cells / metabolism
  • Rats
  • Receptors, Glutamate / metabolism*
  • Recombinant Proteins / metabolism
  • Symporters*
  • Xenopus

Substances

  • Amino Acid Transport System X-AG
  • Excitatory Amino Acid Transporter 4
  • Glutamate Plasma Membrane Transport Proteins
  • Protons
  • Receptors, Glutamate
  • Recombinant Proteins
  • Slc1a6 protein, rat
  • Symporters
  • Arachidonic Acid