Contribution of calcium-activated potassium channels to the vasodilator effect of bradykinin in the isolated, perfused kidney of the rat

Br J Pharmacol. 1996 Jul;118(6):1504-8. doi: 10.1111/j.1476-5381.1996.tb15566.x.

Abstract

1. NO- and prostaglandin-independent, endothelium-dependent vasodilator responses to bradykinin are attributed to release of a hyperpolarizing factor. Therefore, the contribution of K+ channels to the renal vasodilator effect of bradykinin was examined in rat perfused kidneys that were preconstricted with phenylephrine and treated with NG-nitro-L-arginine (L-NOARG) and indomethacin to inhibit NO and prostaglandin synthesis. 2. The non-specific K+ channel inhibitors, TEA and TBA reduced vasodilator responses to bradykinin and cromakalim but not those to nitroprusside. 3. Glibenclamide, an inhibitor of ATP-sensitive K+ channels, blocked the vasodilator response to cromakalim without affecting responses to bradykinin. 4. Charybdotoxin, a selective inhibitor of Ca(2+)-activated K+ channels, greatly attenuated vasodilator responses to bradykinin without affecting those to cromakalim or nitroprusside. 5. Iberiotoxin and leiurotoxin, inhibitors of large and small conductance Ca(2+)-activated K+ channels, respectively, were without effect on vasodilator responses to bradykinin, cromakalim or nitroprusside. 6. These results implicate K+ channels, specifically Ca(2+)-activated K+ channels of intermediate conductance, in the renal vasodilator effect of bradykinin and, thereby, support a role for a hyperpolarizing factor.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenosine Triphosphate / physiology
  • Animals
  • Benzopyrans / pharmacology
  • Bradykinin / pharmacology*
  • Calcium / physiology*
  • Cromakalim
  • Endothelium, Vascular / physiology
  • In Vitro Techniques
  • Kidney / drug effects*
  • Kidney / metabolism
  • Male
  • Nitric Oxide / antagonists & inhibitors
  • Nitric Oxide / physiology
  • Nitroprusside / pharmacology
  • Potassium Channels / drug effects
  • Potassium Channels / physiology*
  • Prostaglandin Antagonists / pharmacology
  • Pyrroles / pharmacology
  • Rats
  • Rats, Wistar
  • Renal Circulation / drug effects
  • Vasodilation / drug effects
  • Vasodilation / physiology*
  • Vasodilator Agents / pharmacology

Substances

  • Benzopyrans
  • Potassium Channels
  • Prostaglandin Antagonists
  • Pyrroles
  • Vasodilator Agents
  • Cromakalim
  • Nitroprusside
  • Nitric Oxide
  • Adenosine Triphosphate
  • Bradykinin
  • Calcium