Lyophilized liposome encapsulated hemoglobin: evaluation of hemodynamic, biochemical, and hematologic responses

Crit Care Med. 1994 Mar;22(3):480-5.

Abstract

Objective: To characterize the hemodynamic, biochemical, and hematologic responses to the administration of the oxygen-carrying fluid lyophilized liposome-encapsulated hemoglobin in the conscious, normovolemic rat.

Design: Prospective, randomized trial.

Setting: Animal laboratory, Jefferson Medical College.

Subjects: Eighty-four male Sprague-Dawley rats.

Interventions: Catheters were introduced into the right atrium (through the jugular vein) and both femoral arteries of test animals, and a thermistor was placed in the ascending aorta through the left common carotid artery for infusion of lyophilized liposome-encapsulated hemoglobin, blood collection, and blood pressure (BP) and cardiac output determinations.

Measurements and main results: Lyophilized liposome-encapsulated hemoglobin (n = 8) infusion (1 mL/min iv) at 1 or 6 mL/kg (10% of estimated blood volume) had no detectable effect on BP, cardiac output, total peripheral resistance, and heart rate during the 5-hr observation period. The infusion also had no effect on hematocrit, leukocyte count, and serum tumor necrosis factor-alpha concentrations. Survival at 7 days was 100% (n = 20). Lyophilized liposome-encapsulated hemoglobin caused transient (2-hr) thrombocytopenia (-24 +/- 9% vs. a Ringer's lactate control group, p < .01), and marginally increased serum thromboxane B2 concentrations (14.6 +/- 6 pg/100 microL, p < .01).

Conclusions: These data suggest that lyophilized liposome-encapsulated hemoglobin can be safely administered to conscious rats, supporting the development of this substance as a potential blood substitute.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • 6-Ketoprostaglandin F1 alpha / blood
  • Animals
  • Drug Carriers
  • Freeze Drying
  • Hemodynamics / drug effects*
  • Hemoglobins / pharmacology*
  • Liposomes
  • Male
  • Prospective Studies
  • Random Allocation
  • Rats
  • Rats, Sprague-Dawley
  • Thromboxane B2 / blood
  • Time Factors
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Drug Carriers
  • Hemoglobins
  • Liposomes
  • Tumor Necrosis Factor-alpha
  • Thromboxane B2
  • 6-Ketoprostaglandin F1 alpha