Effect of Danggui Buxue decoction on hypoxia-induced injury of retinal Müller cells in vitro

Eur J Histochem. 2024 Nov 25;68(4). doi: 10.4081/ejh.2024.4140.

Abstract

Retinopathy is a common complication of diabetes mellitus and the leading cause of visual impairment. Danggui Buxue decoction (RRP) has been used as a traditional drug for the treatment of diabetic nephropathy for many years. The aim of this study was to investigate the effects of RRP on hypoxia-induced retinal Müller cell injury. A model of retinal Müller cell damage was created using high glucose levels (25 mmol/L) and/or exposure to low oxygen conditions (1% O2). RRP was given to rats by continuous gavage for 7 days to obtain drug-containing serum. After sterilization, the serum was added to the culture medium at a ratio of 10%. Cell viability, apoptosis, and cell proliferation were assessed using the CCK-8 kit, Annexin V-FITC/propidium iodide apoptosis kit, and EdU kit. The mRNA levels of angiogenesis factors (ANGPTL4, VEGF) and inflammatory factors (IL-1B, ICAM-1) were detected by RT-qPCR. Western blot analysis was employed to assess the levels of proteins related to the ATF4/CHOP pathway. Following hypoxia for 48 h and 72 h, there was a significant decrease in cell viability and proliferation, as well as a notable increase in apoptosis compared to the control group (21% O2). However, high glucose stimulation had no significant effect, and high glucose combined with hypoxia had no further damage to cells. After 48 h of exposure to low oxygen levels, the mRNA expression levels of ANGPTL4, VEGF, IL-1B, and ICAM-1 in retinal Müller cells were significantly higher than in the control group (21% O2). RRP treatment significantly alleviated the increase of cell apoptosis and the upregulation of IL-1B and-1 in retinal Müller cells induced by hypoxia. RRP has the potential to reduce the suppression of the ATF4/CHOP pathway in hypoxia-induced retinal Müller cells, and it significantly alleviates cell apoptosis through regulating inflammatory factors and the ATF4/CHOP pathway.

MeSH terms

  • Angiopoietin-Like Protein 4 / metabolism
  • Animals
  • Apoptosis* / drug effects
  • Cell Hypoxia / drug effects
  • Cell Proliferation / drug effects
  • Cell Survival / drug effects
  • Cells, Cultured
  • Diabetic Retinopathy / drug therapy
  • Diabetic Retinopathy / metabolism
  • Diabetic Retinopathy / pathology
  • Drugs, Chinese Herbal* / pharmacology
  • Ependymoglial Cells* / drug effects
  • Ependymoglial Cells* / metabolism
  • Ependymoglial Cells* / pathology
  • Intercellular Adhesion Molecule-1 / metabolism
  • Interleukin-1beta / metabolism
  • Male
  • Rats
  • Rats, Sprague-Dawley*
  • Transcription Factor CHOP / metabolism
  • Vascular Endothelial Growth Factor A / metabolism

Substances

  • Drugs, Chinese Herbal
  • danggui buxue decoction
  • ANGPTL4 protein, rat
  • Transcription Factor CHOP
  • Angiopoietin-Like Protein 4
  • Vascular Endothelial Growth Factor A
  • Ddit3 protein, rat
  • vascular endothelial growth factor A, rat
  • Intercellular Adhesion Molecule-1
  • Interleukin-1beta
  • ICAM1 protein, rat