Pullulan dialdehyde cross-linked dual-action adhesive with high adhesion to lung tissue and the capability of pH-responsive drug release

Carbohydr Polym. 2025 Jan 15;348(Pt B):122906. doi: 10.1016/j.carbpol.2024.122906. Epub 2024 Oct 28.

Abstract

To address the main challenges for thoracoscopic lung cancer surgery, including persistent pulmonary air leaks and cancer recurrence, this study developed an in-situ adhesive that can effectively adhere to the lung and release the anticancer drug in response to pH. The adhesive was formulated using hydrophobically modified cold-water fish skin gelatin (hm-CFG) and cross-linking agent pullulan dialdehyde (PDA), in which succinic dihydrazide-modified doxorubicin (SDH-DOX) can be incorporated. Utilizing PDA could improve both cohesion and interfacial adhesion, while also offering drug-loading sites through the aldehyde groups that were not involved in cross-linking. The optimal adhesive formulation was 9C10-CFG/PDA (30 w/v% 9 mol% decanal modified CFG/20 w/v% PDA). The 9C10-CFG/PDA adhesive exhibited suitable cohesive strength, good mechanical flexibility (tensile strain over 170 %), and strong interface adhesion. The burst strength of 9C10-CFG/PDA adhesive (131.5 ± 22.2 mm Hg) was almost 6-fold higher than that of commercial fibrin sealant. In a rat pneumothorax model, 9C10-CFG/PDA adhesive displayed favorable wound-sealing properties, as evidenced by CT imaging and restored rat behavior. When combined with the anticancer drug, SDH-DOX@Adhesive could release the drug in response to pH more gradually than DOX@Adhesive. This dual-action adhesive is anticipated to mitigate post-surgical occurrences of lung air leaks and cancer recurrence.

Keywords: Dual-action adhesive; Hydrophobically modified gelatin; Pullulan dialdehyde; Pulmonary air leak; pH-responsive release.

MeSH terms

  • Adhesives / chemistry
  • Animals
  • Antibiotics, Antineoplastic / administration & dosage
  • Antibiotics, Antineoplastic / chemistry
  • Antibiotics, Antineoplastic / pharmacology
  • Cross-Linking Reagents / chemistry
  • Doxorubicin* / chemistry
  • Doxorubicin* / pharmacology
  • Drug Liberation*
  • Gelatin / chemistry
  • Glucans* / chemistry
  • Humans
  • Hydrogen-Ion Concentration
  • Lung / drug effects
  • Lung / metabolism
  • Lung Neoplasms / drug therapy
  • Male
  • Rats
  • Rats, Sprague-Dawley

Substances

  • pullulan
  • Glucans
  • Doxorubicin
  • Adhesives
  • Gelatin
  • Cross-Linking Reagents
  • Antibiotics, Antineoplastic