HDAC Inhibitors Induce HLA Class I Molecules through the SOX10-IRF1 Axis in Clear Cell Sarcoma Cells

Biol Pharm Bull. 2024;47(11):1913-1919. doi: 10.1248/bpb.b24-00640.

Abstract

Although immune checkpoint inhibitors (ICIs) are an effective treatment for clear cell sarcoma (CCS), a rare melanocytic sarcoma with a poor prognosis, their efficacies are still limited. Therefore, a novel therapeutic strategy is required to improve the efficacy of ICIs. We previously reported that histone deacetylase (HDAC) inhibitors increased melanoma immunogenicity through the SOX10-IRF1 pathway and may improve the efficacy of ICIs for melanoma. We herein demonstrated that the inhibition of HDAC induced the expression of HLA class I molecules through IRF1 in CCS cells, similar to melanoma. The suppression of SOX10 by small interfering RNA (siRNA) induced the expression of HLA class I molecules. In addition, the isoform-specific inhibition of HDAC1/3 induced the expression of another IRF1 downstream molecule, PD-L1 in CCS cells in concert with the suppression of SOX10. Furthermore, the knockdown of IRF1 impaired the induction of PD-L1 expression in CCS cells. Therefore, the inhibition of HDAC1/3 has potential as a novel strategy to increase immunogenicity and as combination therapy with ICIs for CCS and melanoma.

Keywords: IRF1; PD-L1; SOX10; clear cell sarcoma; histone deacetylase inhibitor.

MeSH terms

  • B7-H1 Antigen / metabolism
  • Cell Line, Tumor
  • Histocompatibility Antigens Class I / metabolism
  • Histone Deacetylase 1 / metabolism
  • Histone Deacetylase Inhibitors* / pharmacology
  • Histone Deacetylase Inhibitors* / therapeutic use
  • Histone Deacetylases / metabolism
  • Humans
  • Immune Checkpoint Inhibitors / pharmacology
  • Immune Checkpoint Inhibitors / therapeutic use
  • Interferon Regulatory Factor-1* / genetics
  • Interferon Regulatory Factor-1* / metabolism
  • Melanoma / drug therapy
  • Melanoma / immunology
  • Melanoma / metabolism
  • RNA, Small Interfering
  • SOXE Transcription Factors* / genetics
  • SOXE Transcription Factors* / metabolism
  • Sarcoma, Clear Cell* / drug therapy
  • Sarcoma, Clear Cell* / metabolism

Substances

  • Interferon Regulatory Factor-1
  • Histone Deacetylase Inhibitors
  • SOXE Transcription Factors
  • IRF1 protein, human
  • SOX10 protein, human
  • B7-H1 Antigen
  • CD274 protein, human
  • Histocompatibility Antigens Class I
  • Histone Deacetylases
  • Histone Deacetylase 1
  • histone deacetylase 3
  • HDAC1 protein, human
  • RNA, Small Interfering
  • Immune Checkpoint Inhibitors