Antimicrobial Properties and Therapeutic Potential of Bioactive Compounds in Nigella sativa: A Review

Molecules. 2024 Oct 17;29(20):4914. doi: 10.3390/molecules29204914.

Abstract

Nigella sativa (N. sativa; Ranunculaceae), commonly referred to as black cumin, is one of the most widely used medicinal plants worldwide, with its seeds having numerous applications in the pharmaceutical and food industries. With the emergence of antibiotic resistance in pathogens as an important health challenge, the need for alternative microbe-inhibitory agents is on the rise, whereby black cumin has gained considerable attention from researchers for its strong antimicrobial characteristics owing to its high content in a wide range of bioactive compounds, including thymoquinone, nigellimine, nigellidine, quercetin, and O-cymene. Particularly, thymoquinone increases the levels of antioxidant enzymes that counter oxidative stress in the liver. Additionally, the essential oil in N. sativa seeds effectively inhibits intestinal parasites and shows moderate activity against some bacteria, including Bacillus subtilis and Staphylococcus aureus. Thymoquinone exhibits minimum inhibitory concentrations (MICs) of 8-16 μg/mL against methicillin-resistant Staphylococcus aureus (MRSA) and exhibits MIC 0.25 µg/mL against drug-resistant mycobacteria. Similarly, quercetin shows a MIC of 2 mg/mL against oral pathogens, such as Streptococcus mutans and Lactobacillus acidophilus. Furthermore, endophytic fungi isolated from N. sativa have demonstrated antibacterial activity. Therefore, N. sativa is a valuable medicinal plant with potential for medicinal and food-related applications. In-depth exploration of the corresponding therapeutic potential and scope of industrial application warrants further research.

Keywords: Nigella sativa; antibiotic; antimicrobial; bioactive compounds; medicinal plant; microorganisms; thymoquinone.

Publication types

  • Review

MeSH terms

  • Animals
  • Anti-Bacterial Agents / chemistry
  • Anti-Bacterial Agents / pharmacology
  • Anti-Infective Agents* / chemistry
  • Anti-Infective Agents* / pharmacology
  • Antioxidants / chemistry
  • Antioxidants / pharmacology
  • Bacteria / drug effects
  • Benzoquinones / chemistry
  • Benzoquinones / pharmacology
  • Humans
  • Microbial Sensitivity Tests
  • Nigella sativa* / chemistry
  • Oils, Volatile / chemistry
  • Oils, Volatile / pharmacology
  • Phytochemicals / chemistry
  • Phytochemicals / pharmacology
  • Plant Extracts / chemistry
  • Plant Extracts / pharmacology
  • Plants, Medicinal / chemistry
  • Seeds / chemistry

Substances

  • Anti-Infective Agents
  • Phytochemicals
  • Plant Extracts
  • thymoquinone
  • Antioxidants
  • Benzoquinones
  • Oils, Volatile
  • Anti-Bacterial Agents

Grants and funding

This work is supported by grants from the Intergovernmental International Scientific and Technological Innovation and Cooperation Program of The National Key R&D Program (2023YFE0199200), the National Science Foundation of China (Grant Nos. 32070662 and 32030063), and Joint Research Funds for Medical and Engineering and Scientific Research at Shanghai Jiao Tong University (YG2021ZD02).