The Role and Function of TRPM8 in the Digestive System

Biomolecules. 2024 Jul 21;14(7):877. doi: 10.3390/biom14070877.

Abstract

Transient receptor potential (TRP) melastatin member 8 (TRPM8) is a non-selective cation channel that can be activated by low temperatures (8-26 °C), cooling agents (including menthol analogs such as menthol, icilin, and WS-12), voltage, and extracellular osmotic pressure changes. TRPM8 expression has been identified in the digestive system by several research teams, demonstrating its significant involvement in tissue function and pathologies of the digestive system. Specifically, studies have implicated TRPM8 in various physiological and pathological processes of the esophagus, stomach, colorectal region, liver, and pancreas. This paper aims to comprehensively outline the distinct role of TRPM8 in different organs of the digestive system, offering insights for future mechanistic investigations of TRPM8. Additionally, it presents potential therapeutic targets for treating conditions such as digestive tract inflammation, tumors, sensory and functional disorders, and other related diseases. Furthermore, this paper addresses the limitations of existing studies and highlights the research prospects associated with TRPM8.

Keywords: TRPM8; digestive system; menthol.

Publication types

  • Review

MeSH terms

  • Animals
  • Digestive System / metabolism
  • Humans
  • TRPM Cation Channels* / metabolism

Substances

  • TRPM Cation Channels
  • TRPM8 protein, human

Grants and funding

This research was funded by the National Natural Science Foundation of China grant number 81570490 and 82070555. And The APC was funded by Xiaoyun Yu.