THBS1 and THBS2 Enhance the In Vitro Proliferation, Adhesion, Migration and Invasion of Intrahepatic Cholangiocarcinoma Cells

Int J Mol Sci. 2024 Feb 1;25(3):1782. doi: 10.3390/ijms25031782.

Abstract

In intrahepatic cholangiocarcinoma (iCCA), thrombospondin 1 (THBS1) and 2 (THBS2) are soluble mediators released in the tumor microenvironment (TME) that contribute to the metastatic spreading of iCCA cells via a lymphatic network by the trans-differentiation of vascular endothelial cells to a lymphatic-like phenotype. To study the direct role of THBS1 and THBS2 on the iCCA cells, well-established epithelial (HuCCT-1) and mesenchymal (CCLP1) iCCA cell lines were subjected to recombinant human THBS1 and THBS2 (rhTHBS1, rhTHBS2) for cellular function assays. Cell growth, cell adhesion, migration, and invasion were all enhanced in both CCLP1 and HuCCT-1 cells by the treatment with either rhTHBS1 or rhTHBS2, although they showed some variability in their intensity of speeding up cellular processes. rhTHBS2 was more intense in inducing invasiveness and in committing the HuCCT-1 cells to a mesenchymal-like phenotype and was therefore a stronger enhancer of the malignant behavior of iCCA cells compared to rhTHBS1. Our data extend the role of THBS1 and THBS2, which are not only able to hinder the vascular network and promote tumor-associated lymphangiogenesis but also exacerbate the malignant behavior of the iCCA cells.

Keywords: THBS1; THBS2; angiogenesis; intrahepatic cholangiocarcinoma; lymphangiogenesis; tumor microenvironment.

MeSH terms

  • Bile Duct Neoplasms* / metabolism
  • Bile Ducts, Intrahepatic / metabolism
  • Cell Proliferation / genetics
  • Cholangiocarcinoma* / metabolism
  • Endothelial Cells / metabolism
  • Humans
  • Thrombospondin 1 / genetics
  • Thrombospondin 1 / metabolism
  • Thrombospondins
  • Tumor Microenvironment

Substances

  • Thrombospondin 1
  • thrombospondin 2
  • Thrombospondins

Grants and funding

This work was supported by AMMF—The Cholangiocarcinoma Charity (AMMF Grant Ref: 2022/211), the Next Generation EU—Italian Ministry of University and Research (MUR) PRIN 2022 (Ref: 2022L3BW2P), and Sapienza University of Rome—Fondi di Ateneo (RM12117A0E3970E4; RM122180FA0683A4).