Synthetic Approaches to α-, β-, γ-, and δ-lycoranes

European J Org Chem. 2023 Sep 14;26(35):e202300404. doi: 10.1002/ejoc.202300404. Epub 2023 Jul 11.

Abstract

Lycorane is a pentacyclic core presented in alkaloids isolated from the Amaryllidaceae family of herbaceous flowering plants. Members of this class of natural products have shown to display important biological properties including analgesic, antiviral, and antiproliferative activities. This review presents the known synthetic routes toward α-, β-, γ-, and δ-lycoranes. α-(19 routes), β-(10 routes), γ-(38 routes), and δ-(6 routes).

Keywords: synthesis; α-lycoranes; β-lycoranes; γ-lycoranes; δ-lycoranes.