Long-term outcomes and persistent toxicities following BRAF/MEK inhibitor therapy for advanced melanoma

Eur J Cancer. 2023 Nov:194:113354. doi: 10.1016/j.ejca.2023.113354. Epub 2023 Sep 22.

Abstract

Background: Recent studies have shown that approximately 20% of patients have 4-5 year progression free survival (PFS) on BRAF/MEK inhibitors. The long-term safety and efficacy in these patients with more durable responses have not been studied.

Methods: This retrospective multicenter cohort study assessed response, progression, and adverse events in patients from eight institutions in four countries with >4-year PFS following BRAF/MEK inhibitors.

Results: Among 146 patients, 112 (76.7%) remained progression-free at median follow-up of 7.8 years from treatment start; 131 (89.7%) were alive. Among progressors (n = 34), 21 (62%) were on treatment at progression. Among those who discontinued treatment for reasons other than progression (toxicity, preference, etc.) (n = 68, with median 49 months treatment duration), 13 (19%) progressed (median 15.3 months from treatment cessation to progression). Surgery or radiation for single-organ progression resulted in durable benefit in 11 of 22 patients (50%). Subsequent systemic therapy included immune therapy (24% responded) and BRAF/MEK rechallenge (56% responded). Thirteen (8.9%) patients had ongoing toxicities at last follow-up, 10 (77%) of which remained on active treatment; all cardiac adverse events had resolved (n = 9). Twenty-four (16.4%) patients developed any new primary cancer, and 28 (19%) patients experienced other major health events.

Conclusions: Over 75% of patients with 4-year PFS from BRAF/MEK inhibitors had continued durable antitumor responses after nearly 8-year median follow-up, with similar results in patients who discontinued therapy for reasons other than progression. Long-term toxicities were uncommon and low-grade. These findings highlight the often-favourable outcomes in patients with extended benefit from BRAF/MEK inhibitors.

Keywords: Adverse events; BRAF/MEK inhibitors; Melanoma; Targeted therapy.

Publication types

  • Multicenter Study
  • Research Support, Non-U.S. Gov't
  • Research Support, N.I.H., Extramural

MeSH terms

  • Antineoplastic Combined Chemotherapy Protocols / adverse effects
  • Cohort Studies
  • Humans
  • Melanoma* / pathology
  • Mitogen-Activated Protein Kinase Kinases
  • Mutation
  • Protein Kinase Inhibitors / adverse effects
  • Proto-Oncogene Proteins B-raf / genetics
  • Skin Neoplasms* / pathology

Substances

  • Proto-Oncogene Proteins B-raf
  • Protein Kinase Inhibitors
  • Mitogen-Activated Protein Kinase Kinases
  • BRAF protein, human