Evaluating the Performance of Pathogen-Targeted Positron Emission Tomography Radiotracers in a Rat Model of Vertebral Discitis-Osteomyelitis

J Infect Dis. 2023 Oct 3;228(Suppl 4):S281-S290. doi: 10.1093/infdis/jiad159.

Abstract

Background: Vertebral discitis-osteomyelitis (VDO) is a devastating infection of the spine that is challenging to distinguish from noninfectious mimics using computed tomography and magnetic resonance imaging. We and others have developed novel metabolism-targeted positron emission tomography (PET) radiotracers for detecting living Staphylococcus aureus and other bacteria in vivo, but their head-to-head performance in a well-validated VDO animal model has not been reported.

Methods: We compared the performance of several PET radiotracers in a rat model of VDO. [11C]PABA and [18F]FDS were assessed for their ability to distinguish S aureus, the most common non-tuberculous pathogen VDO, from Escherichia coli.

Results: In the rat S aureus VDO model, [11C]PABA could detect as few as 103 bacteria and exhibited the highest signal-to-background ratio, with a 20-fold increased signal in VDO compared to uninfected tissues. In a proof-of-concept experiment, detection of bacterial infection and discrimination between S aureus and E coli was possible using a combination of [11C]PABA and [18F]FDS.

Conclusions: Our work reveals that several bacteria-targeted PET radiotracers had sufficient signal to background in a rat model of S aureus VDO to be potentially clinically useful. [11C]PABA was the most promising tracer investigated and warrants further investigation in human VDO.

Keywords: S aureus; Infection imaging; metabolism; nuclear medicine; positron emission tomography.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, N.I.H., Extramural

MeSH terms

  • 4-Aminobenzoic Acid
  • Animals
  • Bacteria
  • Discitis* / diagnostic imaging
  • Escherichia coli
  • Humans
  • Osteomyelitis* / microbiology
  • Positron-Emission Tomography / methods
  • Radiopharmaceuticals
  • Rats
  • Staphylococcal Infections* / diagnostic imaging
  • Staphylococcus aureus

Substances

  • Carbon-11
  • 4-Aminobenzoic Acid
  • Radiopharmaceuticals