Nucleoside diphosphate kinases 1 and 2 regulate a protective liver response to a high-fat diet

Sci Adv. 2023 Sep 8;9(36):eadh0140. doi: 10.1126/sciadv.adh0140. Epub 2023 Sep 6.

Abstract

The synthesis of fatty acids from acetyl-coenzyme A (AcCoA) is deregulated in diverse pathologies, including cancer. Here, we report that fatty acid accumulation is negatively regulated by nucleoside diphosphate kinases 1 and 2 (NME1/2), housekeeping enzymes involved in nucleotide homeostasis that were recently found to bind CoA. We show that NME1 additionally binds AcCoA and that ligand recognition involves a unique binding mode dependent on the CoA/AcCoA 3' phosphate. We report that Nme2 knockout mice fed a high-fat diet (HFD) exhibit excessive triglyceride synthesis and liver steatosis. In liver cells, NME2 mediates a gene transcriptional response to HFD leading to the repression of fatty acid accumulation and activation of a protective gene expression program via targeted histone acetylation. Our findings implicate NME1/2 in the epigenetic regulation of a protective liver response to HFD and suggest a potential role in controlling AcCoA usage between the competing paths of histone acetylation and fatty acid synthesis.

MeSH terms

  • Animals
  • Diet, High-Fat / adverse effects
  • Epigenesis, Genetic
  • Fatty Acids
  • Histones
  • Liver
  • Mice
  • Mice, Knockout
  • Nucleoside-Diphosphate Kinase* / genetics

Substances

  • Nucleoside-Diphosphate Kinase
  • Histones
  • Fatty Acids