HER2-Positive Gastric Cancer: The Role of Immunotherapy and Novel Therapeutic Strategies

Int J Mol Sci. 2023 Jul 13;24(14):11403. doi: 10.3390/ijms241411403.

Abstract

Gastric cancer is an aggressive disease with increasing global incidence in recent years. Human epidermal growth receptor 2 (HER2) is overexpressed in approximately 10-20% of gastric cancers. The implementation of targeted therapy against HER2 as part of the standard of care treatment in metastatic disease has improved the prognosis of this subset of patients. However, gastric cancer still has high mortality rates and urgently requires new treatment strategies. The combination of immunotherapy with HER2-targeted therapies has shown synergistic effects in preclinical models, this being the rationale behind exploring this combination in clinical trials in locally advanced and metastatic settings. Additionally, the irruption of antibody-drug conjugates and other novel HER2-targeted agents has led to the development of numerous clinical trials showing promising results. This review presents the molecular mechanisms supporting the use of HER2-targeted drugs in combination with immunotherapy and provides an overview of the therapeutic scenario of HER2-positive disease. We focus on the role of immunotherapy but also summarize emerging therapies and combinations under clinical research that may change the standard treatment in HER-2 positive disease in the future.

Keywords: HER2; PD-1/PD-L1; antibody-drug conjugate; chemotherapy; clinical trials; gastric cancer; immunotherapy; novel therapies; trastuzumab.

Publication types

  • Review

MeSH terms

  • Antineoplastic Agents* / pharmacology
  • Antineoplastic Agents* / therapeutic use
  • Humans
  • Immunoconjugates* / therapeutic use
  • Immunotherapy
  • Receptor, ErbB-2* / antagonists & inhibitors
  • Stomach Neoplasms* / drug therapy
  • Trastuzumab / pharmacology
  • Trastuzumab / therapeutic use

Substances

  • Antineoplastic Agents
  • Immunoconjugates
  • Receptor, ErbB-2
  • Trastuzumab

Grants and funding

This research received no external funding.