ACE2 expression and spike S1 protein-mediated immune responses in oral mucosal cells

Oral Dis. 2024 May;30(4):2293-2305. doi: 10.1111/odi.14670. Epub 2023 Jul 19.

Abstract

Objectives: ACE2, known as a host receptor involved with SARS-CoV-2 infection, binds to viral spike proteins for host cell entry. However, details regarding its induction and function in oral mucosal cells remain unknown.

Materials and methods: We examined ACE2 expression and its induction by transfected mimic nucleotides and pro-inflammatory cytokines in oral keratinocytes (RT7) and fibroblasts (GT1). Subsequently, the effects of viral spike S1 protein via ACE2 on CXCL10 expression induced by pro-inflammatory cytokines in both cells were examined.

Results: ACE2 was constitutively expressed in RT7 and GT1. Transfected Poly(I:C) and Poly(dA:dT) increased ACE2 expression in those cells, while knockdown of RIG-I decreased ACE2 expression induced by those transfected ds nucleotides. IFN-γ and TNF-α enhanced transfected ds nucleotides-induced ACE2 expression in RT7 but not GT1. S1 protein alone did not affect CXCL10 expression in either cell type, whereas it enhanced IFN-β-induced CXCL10 in both, while immune responses of IFN-γ- and TNF-α-induced CXCL10 enhanced by S1 protein were different between RT7 and GT1. Finally, knockdown of ACE2 decreased cytokines and S1 protein mediated-CXCL10 levels in both cells.

Conclusions: ACE2 in oral mucosal cells may contribute to development of infection and inflammation in cooperation with pro-inflammatory cytokines following SARS-CoV-2 invasion.

Keywords: ACE2; oral fibroblasts; oral keratinocytes; spike S1 protein.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Angiotensin-Converting Enzyme 2* / genetics
  • Angiotensin-Converting Enzyme 2* / metabolism
  • Cell Line
  • Chemokine CXCL10* / metabolism
  • Cytokines / metabolism
  • Fibroblasts / immunology
  • Fibroblasts / metabolism
  • Humans
  • Keratinocytes* / immunology
  • Keratinocytes* / metabolism
  • Mouth Mucosa* / immunology
  • SARS-CoV-2
  • Spike Glycoprotein, Coronavirus* / immunology
  • Spike Glycoprotein, Coronavirus* / metabolism
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Angiotensin-Converting Enzyme 2
  • Spike Glycoprotein, Coronavirus
  • Chemokine CXCL10
  • spike protein, SARS-CoV-2
  • ACE2 protein, human
  • CXCL10 protein, human
  • Cytokines
  • Tumor Necrosis Factor-alpha