Unlike RNA-TBA (rTBA), iso-rTBA, the 2'-5'-linked RNA-thrombin-binding aptamer, is a functional equivalent of TBA

Chem Commun (Camb). 2023 Feb 2;59(11):1461-1464. doi: 10.1039/d2cc05718b.

Abstract

An antiparallel, functional RNA G-quadruplex of the 2'-5'-linked thrombin-binding aptamer (iso-rTBA) is reported for the first time. It can inhibit clotting and is remarkably stable to nuclease-degradation, besides having high thermal stability. It is thus, a superior candidate to TBA, rTBA or isoTBA, for further development as an anticoagulant.

MeSH terms

  • Anticoagulants / pharmacology
  • Aptamers, Nucleotide* / pharmacology
  • Blood Coagulation
  • G-Quadruplexes*
  • RNA
  • Thrombin

Substances

  • thrombin aptamer
  • RNA
  • Anticoagulants
  • Aptamers, Nucleotide
  • Thrombin