COVID-19 Molecular Pathophysiology: Acetylation of Repurposing Drugs

Int J Mol Sci. 2022 Oct 31;23(21):13260. doi: 10.3390/ijms232113260.

Abstract

Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) induces immune-mediated type 1 interferon (IFN-1) production, the pathophysiology of which involves sterile alpha motif and histidine-aspartate domain-containing protein 1 (SAMHD1) tetramerization and the cytosolic DNA sensor cyclic-GMP-AMP synthase (cGAS)-stimulator of interferon genes (STING) signaling pathway. As a result, type I interferonopathies are exacerbated. Aspirin inhibits cGAS-mediated signaling through cGAS acetylation. Acetylation contributes to cGAS activity control and activates IFN-1 production and nuclear factor-κB (NF-κB) signaling via STING. Aspirin and dapsone inhibit the activation of both IFN-1 and NF-κB by targeting cGAS. We define these as anticatalytic mechanisms. It is necessary to alleviate the pathologic course and take the lag time of the odds of achieving viral clearance by day 7 to coordinate innate or adaptive immune cell reactions.

Keywords: ACE2 (angiotensin-converting enzyme 2); SAMHD1 (sterile alpha motif and histidine-aspartate domain-containing protein 1); SARS-CoV-2 (severe acute respiratory syndrome coronavirus 2); TLR4 (Toll-like receptor 4); aspirin; cGAS–STING (cyclic guanosine monophosphate (GMP)-adenosine monophosphate (AMP) synthase (cGAS)–stimulator of interferon genes (STING)); dapsone; dexamethasone; immunologic engram; inflammasome; spike protein.

Publication types

  • Review

MeSH terms

  • Acetylation
  • Aspirin
  • COVID-19 Drug Treatment*
  • Drug Repositioning
  • Humans
  • Immunity, Innate / genetics
  • Interferon Type I* / metabolism
  • Membrane Proteins / metabolism
  • NF-kappa B / metabolism
  • Nucleotidyltransferases / metabolism
  • SARS-CoV-2

Substances

  • NF-kappa B
  • Membrane Proteins
  • Nucleotidyltransferases
  • Interferon Type I
  • Aspirin

Grants and funding

This research received no external funding.