NIMA-related kinase 9 regulates the phosphorylation of the essential myosin light chain in the heart

Nat Commun. 2022 Oct 20;13(1):6209. doi: 10.1038/s41467-022-33658-2.

Abstract

To adapt to changing hemodynamic demands, regulatory mechanisms modulate actin-myosin-kinetics by calcium-dependent and -independent mechanisms. We investigate the posttranslational modification of human essential myosin light chain (ELC) and identify NIMA-related kinase 9 (NEK9) to interact with ELC. NEK9 is highly expressed in the heart and the interaction with ELC is calcium-dependent. Silencing of NEK9 results in blunting of calcium-dependent ELC-phosphorylation. CRISPR/Cas9-mediated disruption of NEK9 leads to cardiomyopathy in zebrafish. Binding to ELC is mediated via the protein kinase domain of NEK9. A causal relationship between NEK9 activity and ELC-phosphorylation is demonstrated by genetic sensitizing in-vivo. Finally, we observe significantly upregulated ELC-phosphorylation in dilated cardiomyopathy patients and provide a unique map of human ELC-phosphorylation-sites. In summary, NEK9-mediated ELC-phosphorylation is a calcium-dependent regulatory system mediating cardiac contraction and inotropy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Actins* / metabolism
  • Animals
  • Calcium / metabolism
  • Humans
  • Myosin Light Chains* / metabolism
  • NIMA-Related Kinases / genetics
  • NIMA-Related Kinases / metabolism
  • Phosphorylation
  • Protein Kinases / metabolism
  • Zebrafish / metabolism

Substances

  • Myosin Light Chains
  • Actins
  • Calcium
  • NIMA-Related Kinases
  • Protein Kinases
  • NEK9 protein, human