Signaling through Free Fatty Acid Receptor 4 Attenuates Cardiometabolic Disease

Physiology (Bethesda). 2022 Nov 1;37(6):311-322. doi: 10.1152/physiol.00007.2022. Epub 2022 Aug 9.

Abstract

A surge in the prevalence of obesity and metabolic syndrome, which promote systemic inflammation, underlies an increase in cardiometabolic disease. Free fatty acid receptor 4 is a nutrient sensor for long-chain fatty acids, like ω3-polyunsaturated fatty acids (ω3-PUFAs), that attenuates metabolic disease and resolves inflammation. Clinical trials indicate ω3-PUFAs are cardioprotective, and this review discusses the mechanistic links between ω3-PUFAs, free fatty acid receptor 4, and attenuation of cardiometabolic disease.

Keywords: 18-hydroxyeicosapentaenoic acid (18-HEPE); cardiometabolic disease; free fatty acid receptor 4 (Ffar4); heart; specialized proresolving mediators (SPM); ω3-polyunsaturated fatty acids (ω3-PUFAs).

Publication types

  • Review
  • Research Support, N.I.H., Extramural

MeSH terms

  • Cardiovascular Diseases*
  • Fatty Acids, Nonesterified
  • Fatty Acids, Omega-3* / metabolism
  • Fatty Acids, Omega-3* / therapeutic use
  • Humans
  • Inflammation
  • Signal Transduction

Substances

  • Fatty Acids, Nonesterified
  • Fatty Acids, Omega-3