Radical Perfluoroalkylation of Arenes via Carbanion Intermediates

J Org Chem. 2021 Aug 6;86(15):10903-10913. doi: 10.1021/acs.joc.1c01296. Epub 2021 Jul 21.

Abstract

The use of sodium dithionite with perfluoroalkyl iodides under basic conditions facilitates the direct perfluoroalkylation of arenes with pendant benzylic electron-withdrawing groups. This occurs via attack of the arene on the electrophilic perfluoroalkyl radical, through the donation of electron density from a benzylic anion. The substrate scope was expanded beyond benzylic nitriles with cyclic substrates bearing electron-withdrawing groups at the benzylic position-enforcing donation of electron density to the aromatic ring and enabling attack on the perfluoroalkyl radical.

MeSH terms

  • Electrons
  • Iodides*
  • Molecular Structure
  • Nitriles*

Substances

  • Iodides
  • Nitriles