Solvent-Minimized Synthesis of 4CzIPN and Related Organic Fluorophores via Ball Milling

J Org Chem. 2021 Oct 15;86(20):14095-14101. doi: 10.1021/acs.joc.1c01233. Epub 2021 Jul 14.

Abstract

The mechanochemical synthesis of 2,4,5,6-tetra(9H-carbazol-9-yl)isophthalonitrile and related organic fluorophores/photocatalysts via a solvent-minimized four-fold SNAr pathway is herein described. Employing sodium tert-butoxide as base, and negating the need for any air/moisture-sensitive reaction set-ups, a selection of organic dyes was synthesized in just 1 h using this ball-milling technique. Furthermore, the transformation was then showcased on a multigram scale.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Ionophores
  • Solvents*

Substances

  • Ionophores
  • Solvents