A unique subset of glycolytic tumour-propagating cells drives squamous cell carcinoma

Nat Metab. 2021 Feb;3(2):182-195. doi: 10.1038/s42255-021-00350-6. Epub 2021 Feb 22.

Abstract

Head and neck squamous cell carcinoma (SCC) remains among the most aggressive human cancers. Tumour progression and aggressiveness in SCC are largely driven by tumour-propagating cells (TPCs). Aerobic glycolysis, also known as the Warburg effect, is a characteristic of many cancers; however, whether this adaptation is functionally important in SCC, and at which stage, remains poorly understood. Here, we show that the NAD+-dependent histone deacetylase sirtuin 6 is a robust tumour suppressor in SCC, acting as a modulator of glycolysis in these tumours. Remarkably, rather than a late adaptation, we find enhanced glycolysis specifically in TPCs. More importantly, using single-cell RNA sequencing of TPCs, we identify a subset of TPCs with higher glycolysis and enhanced pentose phosphate pathway and glutathione metabolism, characteristics that are strongly associated with a better antioxidant response. Together, our studies uncover enhanced glycolysis as a main driver in SCC, and, more importantly, identify a subset of TPCs as the cell of origin for the Warburg effect, defining metabolism as a key feature of intra-tumour heterogeneity.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Antioxidants / metabolism
  • Disease Progression
  • Glutathione / metabolism
  • Glycolysis*
  • Head and Neck Neoplasms / pathology*
  • Humans
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Neoplastic Stem Cells / pathology*
  • Pentose Phosphate Pathway
  • RNA, Neoplasm / genetics
  • Single-Cell Analysis
  • Sirtuins / genetics
  • Sirtuins / metabolism
  • Squamous Cell Carcinoma of Head and Neck / pathology*
  • Xenograft Model Antitumor Assays

Substances

  • Antioxidants
  • RNA, Neoplasm
  • Sirt6 protein, mouse
  • SIRT6 protein, human
  • Sirtuins
  • Glutathione