Nutraceutical delivery through nano-emulsions: General aspects, recent applications and patented inventions

Colloids Surf B Biointerfaces. 2021 Apr:200:111526. doi: 10.1016/j.colsurfb.2020.111526. Epub 2021 Jan 14.

Abstract

Nanostructured emulsions have a significant potential for encasing, transport and delivery of hydrophilic and lipophilic nutraceuticals and other bioactive compounds by providing enhanced stability and functionality in food and pharmaceutical applications. As highlighted in recent researches, essential fatty acids (EFA) and oils (EO), antioxidants, vitamins, minerals, pro and prebiotics, and co-enzymes, are common bioactives encapsulated in nanoscale delivery systems in order to protect them from degradation during processing and storage, and to improve bioavailability after their consumption. Nanoemulsions (NEs) as delivery systems for nutraceuticals comprise either oil-in-water (O/W) or water-in-oil (W/O) biphasic dispersion with nano-sized droplets, which are stabilized through an active surfactant. Both high- and low- energy methods are used to produce well-structured and stable NEs with advanced structural and rheological features. The in vitro and in vivo studies are focused to assess the nutraceutical releasing profile, gastrointestinal transportation and cytotoxicity of nutraceutical loaded NE. Within the last three decades, a number of NE systems have been developed for certain purposes and submitted for patent approval. Currently, there are many issued patents published as well as and applications under process. This review focus on the current status of food-grade NEs in terms of formation, characterization, relevant applications of nutraceutical delivery, and the recent developments including patented systems.

Keywords: Characterization; Fabrication; Nanoemulsion; Nutraceutical delivery; Patents; Safety.

Publication types

  • Review

MeSH terms

  • Biological Availability
  • Dietary Supplements*
  • Emulsions
  • Inventions*
  • Oils
  • Particle Size

Substances

  • Emulsions
  • Oils