Potential Antiviral Options against SARS-CoV-2 Infection

Viruses. 2020 Jun 13;12(6):642. doi: 10.3390/v12060642.

Abstract

As of June 2020, the number of people infected with severe acute respiratory coronavirus 2 (SARS-CoV-2) continues to skyrocket, with more than 6.7 million cases worldwide. Both the World Health Organization (WHO) and United Nations (UN) has highlighted the need for better control of SARS-CoV-2 infections. However, developing novel virus-specific vaccines, monoclonal antibodies and antiviral drugs against SARS-CoV-2 can be time-consuming and costly. Convalescent sera and safe-in-man broad-spectrum antivirals (BSAAs) are readily available treatment options. Here, we developed a neutralization assay using SARS-CoV-2 strain and Vero-E6 cells. We identified the most potent sera from recovered patients for the treatment of SARS-CoV-2-infected patients. We also screened 136 safe-in-man broad-spectrum antivirals against the SARS-CoV-2 infection in Vero-E6 cells and identified nelfinavir, salinomycin, amodiaquine, obatoclax, emetine and homoharringtonine. We found that a combination of orally available virus-directed nelfinavir and host-directed amodiaquine exhibited the highest synergy. Finally, we developed a website to disseminate the knowledge on available and emerging treatments of COVID-19.

Keywords: antiviral drug combinations; antivirals; broad-spectrum antivirals.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amodiaquine / pharmacology
  • Animals
  • Antiviral Agents / pharmacology*
  • Betacoronavirus / drug effects*
  • COVID-19
  • COVID-19 Serotherapy
  • Caco-2 Cells
  • Cell Line, Tumor
  • Chlorocebus aethiops
  • Coronavirus Infections / drug therapy*
  • Coronavirus Infections / therapy
  • Drug Therapy, Combination
  • Emetine / pharmacology
  • HEK293 Cells
  • HT29 Cells
  • Homoharringtonine / pharmacology
  • Humans
  • Immune Sera / immunology
  • Immunization, Passive / methods
  • Indoles
  • Nelfinavir / pharmacology
  • Neutralization Tests / methods*
  • Pandemics
  • Pneumonia, Viral / drug therapy*
  • Pyrans / pharmacology
  • Pyrroles / pharmacology
  • SARS-CoV-2
  • Vero Cells

Substances

  • Antiviral Agents
  • Immune Sera
  • Indoles
  • Pyrans
  • Pyrroles
  • Amodiaquine
  • salinomycin
  • Homoharringtonine
  • Nelfinavir
  • obatoclax
  • Emetine