Mucosal Profiling of Pediatric-Onset Colitis and IBD Reveals Common Pathogenics and Therapeutic Pathways

Cell. 2019 Nov 14;179(5):1160-1176.e24. doi: 10.1016/j.cell.2019.10.027.

Abstract

Pediatric-onset colitis and inflammatory bowel disease (IBD) have significant effects on the growth of infants and children, but the etiopathogenesis underlying disease subtypes remains incompletely understood. Here, we report single-cell clustering, immune phenotyping, and risk gene analysis for children with undifferentiated colitis, Crohn's disease, and ulcerative colitis. We demonstrate disease-specific characteristics, as well as common pathogenesis marked by impaired cyclic AMP (cAMP)-response signaling. Specifically, infiltration of PDE4B- and TNF-expressing macrophages, decreased abundance of CD39-expressing intraepithelial T cells, and platelet aggregation and release of 5-hydroxytryptamine at the colonic mucosae were common in colitis and IBD patients. Targeting these pathways by using the phosphodiesterase inhibitor dipyridamole restored immune homeostasis and improved colitis symptoms in a pilot study. In summary, comprehensive analysis of the colonic mucosae has uncovered common pathogenesis and therapeutic targets for children with colitis and IBD.

Keywords: CASP7; CD39; PDE4B; TNF; cAMP; dipyridamole; pediatric-onset colitis and IBD; platelet; risk genes; single-cell RNA expression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antigens, CD / metabolism
  • Apyrase / metabolism
  • B-Lymphocytes / drug effects
  • B-Lymphocytes / immunology
  • Cell Death / drug effects
  • Cellular Microenvironment / drug effects
  • Child
  • Cohort Studies
  • Colon / pathology
  • Dendritic Cells / drug effects
  • Dendritic Cells / metabolism
  • Dipyridamole / pharmacology
  • Endothelial Cells / drug effects
  • Endothelial Cells / metabolism
  • Epithelial Cells / drug effects
  • Epithelial Cells / metabolism
  • Epithelial Cells / pathology
  • Fibroblasts / drug effects
  • Fibroblasts / metabolism
  • Gene Expression Regulation / drug effects
  • Genetic Predisposition to Disease
  • Homeostasis / drug effects
  • Humans
  • Immunoglobulin G / blood
  • Immunologic Memory
  • Inflammation / pathology
  • Inflammatory Bowel Diseases / blood
  • Inflammatory Bowel Diseases / genetics
  • Inflammatory Bowel Diseases / pathology*
  • Inflammatory Bowel Diseases / therapy*
  • Interferon Type I / metabolism
  • Intestinal Mucosa / pathology*
  • Macrophages / drug effects
  • Macrophages / metabolism
  • Methylprednisolone / pharmacology
  • Myeloid Cells / drug effects
  • Myeloid Cells / metabolism

Substances

  • Antigens, CD
  • Immunoglobulin G
  • Interferon Type I
  • Dipyridamole
  • Apyrase
  • CD39 antigen
  • Methylprednisolone