Genotoxic stress-triggered β-catenin/JDP2/PRMT5 complex facilitates reestablishing glutathione homeostasis

Nat Commun. 2019 Aug 21;10(1):3761. doi: 10.1038/s41467-019-11696-7.

Abstract

The mechanisms underlying how cells subjected to genotoxic stress reestablish reduction-oxidation (redox) homeostasis to scavenge genotoxic stress-induced reactive oxygen species (ROS), which maintains the physiological function of cellular processes and cell survival, remain unclear. Herein, we report that, via a TCF-independent mechanism, genotoxic stress induces the enrichment of β-catenin in chromatin, where it forms a complex with ATM phosphorylated-JDP2 and PRMT5. This elicits histone H3R2me1/H3R2me2s-induced transcriptional activation by the recruitment of the WDR5/MLL methyltransferase complexes and concomitant H3K4 methylation at the promoters of multiple genes in GSH-metabolic cascade. Treatment with OICR-9429, a small-molecule antagonist of the WDR5-MLL interaction, inhibits the β-catenin/JDP2/PRMT5 complex-reestablished GSH metabolism, leading to a lethal increase in the already-elevated levels of ROS in the genotoxic-agent treated cancer cells. Therefore, our results unveil a plausible role for β-catenin in reestablishing redox homeostasis upon genotoxic stress and shed light on the mechanisms of inducible chemotherapy resistance in cancer.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • A549 Cells
  • Animals
  • Biphenyl Compounds / pharmacology
  • Cell Line, Tumor
  • Chromatin
  • DNA Damage / physiology*
  • Dihydropyridines / pharmacology
  • Female
  • Glutathione / drug effects
  • Glutathione / metabolism*
  • Histone-Lysine N-Methyltransferase / metabolism
  • Histones / metabolism
  • Homeostasis
  • Humans
  • Mice
  • Mice, Inbred NOD
  • Mice, SCID
  • Myeloid-Lymphoid Leukemia Protein / metabolism
  • Neoplasms / metabolism
  • Promoter Regions, Genetic
  • Protein Interaction Domains and Motifs / drug effects
  • Protein-Arginine N-Methyltransferases / metabolism*
  • Reactive Oxygen Species / metabolism
  • Repressor Proteins / metabolism*
  • Transcriptional Activation
  • beta Catenin / metabolism*

Substances

  • Biphenyl Compounds
  • Chromatin
  • Dihydropyridines
  • Histones
  • Jundp2 protein, mouse
  • OICR-9429
  • Reactive Oxygen Species
  • Repressor Proteins
  • beta Catenin
  • Myeloid-Lymphoid Leukemia Protein
  • Prmt5 protein, mouse
  • Protein-Arginine N-Methyltransferases
  • Histone-Lysine N-Methyltransferase
  • Kmt2a protein, mouse
  • Glutathione