Novel strategies for anti-aging drug discovery

Expert Opin Drug Discov. 2017 Sep;12(9):955-966. doi: 10.1080/17460441.2017.1349750. Epub 2017 Jul 11.

Abstract

Scientific achievements in the last few decades, leading to effective therapeutic interventions, have dramatically improved human life expectancy. Consequently, aging has become a significant problem and represents the major risk factor for most human pathologies including diabetes, cardiovascular diseases, neurological disorders, and cancer. Scientific discoveries over the past two decades have been instrumental in dissecting molecular mechanism(s) which play important roles in determining longevity. The same understanding has also led to the acknowledgement of the plurality of 'causes' which act either alone or in combination to create the condition which can be defined as 'aging'. Areas covered: Over the years, several concepts have been put forward for the development of a viable anti-aging regimen. In this review, the authors extensively review anti aging interventions based on caloric restriction, activation of telomerase, autophagy inducers, senolytic therapeutics, plasma membrane redox system (PMRS) activators, epigenetic modulators, and stem cell therapies. Expert opinion: Based upon our current understanding, one of the most promising approaches for a successful anti-aging strategy includes the activation of adenosine monophosphate dependent protein kinase (AMPK). Another strategy may involve activation of PMRS. Future research efforts are likely to focus on nutrient and energy sensing molecular pathways which include mTOR, IGF-1, AMPK and the sirtuins.

Keywords: Anti-aging; PMRS activators; autophagy inducers; caloric restriction; epigenetic modulators; senolytic therapeutics; telomerase activation.

Publication types

  • Review
  • Research Support, Non-U.S. Gov't

MeSH terms

  • AMP-Activated Protein Kinases / metabolism
  • Age Factors
  • Aging / drug effects*
  • Animals
  • Cell Membrane / metabolism
  • Drug Design*
  • Drug Discovery / methods*
  • Humans
  • Longevity / physiology
  • Oxidation-Reduction / drug effects

Substances

  • AMP-Activated Protein Kinases