Effects of histatin-1 peptide on human corneal epithelial cells

PLoS One. 2017 May 23;12(5):e0178030. doi: 10.1371/journal.pone.0178030. eCollection 2017.

Abstract

Purpose: Ocular surface and corneal epithelial wounds are common and potentially debilitating problems. Ideal treatments for these injuries would promote epithelial healing without inflammation, infection and scarring. In addition the best treatments would be cost-efficient, effective, non-toxic and easily applied. Histatin-1 peptides have been shown to be safe and effective enhancers of epithelial wound healing in other model systems. We sought to determine whether histatin-1 peptides could enhance human corneal epithelial wound healing in vitro.

Methods: Histatin-1 peptides were applied to human corneal epithelial cells and compared over useful dose ranges in scratch assays using time-lapse microscopy. In addition, path finding analysis, cell spreading assays, toxicity and proliferation assays were performed to further characterize the effects of histatin-1 peptide on human corneal limbal epithelial (HCLE).

Results: Histatin-1 enhanced human corneal epithelial wound healing in typical wound healing models. There was minimal toxicity and no significant enhancement of proliferation of corneal epithelium in response to histatin-1 application. Corneal epithelial spreading and pathfinding appeared to be enhanced by the application of histatin-1 peptides.

Conclusions: Histatin -1 peptide may enhance migration of HCLE cells and wound healing in vitro. These peptides may have benefit in corneal epithelial wounds and need to be investigated further.

MeSH terms

  • Analysis of Variance
  • Bromodeoxyuridine
  • Cell Movement / drug effects
  • Cell Movement / physiology
  • Cell Proliferation / drug effects
  • Cell Proliferation / physiology
  • Cells, Cultured
  • Corneal Injuries / drug therapy*
  • Corneal Injuries / metabolism
  • Corneal Injuries / pathology
  • Dose-Response Relationship, Drug
  • Drug Evaluation, Preclinical
  • Epithelium, Corneal / drug effects*
  • Epithelium, Corneal / metabolism
  • Epithelium, Corneal / pathology
  • Fluorescent Antibody Technique
  • Histatins / chemical synthesis
  • Histatins / pharmacology*
  • Histatins / toxicity
  • Humans
  • Protective Agents / chemical synthesis
  • Protective Agents / pharmacology*
  • Protective Agents / toxicity
  • Re-Epithelialization / drug effects*
  • Re-Epithelialization / physiology

Substances

  • Histatins
  • Protective Agents
  • Bromodeoxyuridine