Activating MAPK1 (ERK2) mutation in an aggressive case of disseminated juvenile xanthogranuloma

Oncotarget. 2017 Jul 11;8(28):46065-46070. doi: 10.18632/oncotarget.17521.

Abstract

Juvenile xanthogranuloma (JXG) is a rare histiocytic disorder that is usually benign and self-limiting. We present a case of atypical, aggressive JXG harboring a novel mitogen-activated protein kinase (MAPK) pathway mutation in the MAPK1 gene, which encodes mitogen-activated protein kinase 1 or extracellular signal-regulated 2 (ERK2). Our analysis revealed that the mutation results in constitutive ERK activation that is resistant to BRAF or MEK inhibitors but susceptible to an ERK inhibitor. These data highlight the importance of identifying specific MAPK pathway alterations as part of the diagnostic workup for patients with histiocytic disorders rather than initiating empiric treatment with MEK inhibitors.

Keywords: ERK activation; MAPK1; histiocytic disorder; juvenile xanthogranuloma; somatic mutation.

Publication types

  • Case Reports

MeSH terms

  • Cells, Cultured
  • Child
  • Drug Therapy
  • Histiocytes / pathology*
  • Humans
  • Lymph Nodes / pathology
  • Lymph Nodes / physiology*
  • Male
  • Mitogen-Activated Protein Kinase 1 / genetics*
  • Remission Induction
  • Signal Transduction / genetics
  • Stem Cell Transplantation
  • Xanthogranuloma, Juvenile / diagnosis
  • Xanthogranuloma, Juvenile / genetics*

Substances

  • MAPK1 protein, human
  • Mitogen-Activated Protein Kinase 1