Steviol glycosides enhance pancreatic beta-cell function and taste sensation by potentiation of TRPM5 channel activity

Nat Commun. 2017 Mar 31:8:14733. doi: 10.1038/ncomms14733.

Abstract

Steviol glycosides (SGs), such as stevioside and rebaudioside A, are natural, non-caloric sweet-tasting organic molecules, present in extracts of the scrub plant Stevia rebaudiana, which are widely used as sweeteners in consumer foods and beverages. TRPM5 is a Ca2+-activated cation channel expressed in type II taste receptor cells and pancreatic β-cells. Here we show that stevioside, rebaudioside A and their aglycon steviol potentiate the activity of TRPM5. We find that SGs potentiate perception of bitter, sweet and umami taste, and enhance glucose-induced insulin secretion in a Trpm5-dependent manner. Daily consumption of stevioside prevents development of high-fat-diet-induced diabetic hyperglycaemia in wild-type mice, but not in Trpm5-/- mice. These results elucidate a molecular mechanism of action of SGs and identify TRPM5 as a potential target to prevent and treat type 2 diabetes.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blood Glucose / drug effects
  • Blood Glucose / metabolism
  • Diabetes Mellitus, Type 2 / metabolism
  • Diet, High-Fat
  • Diterpenes, Kaurane / pharmacology*
  • Female
  • Glucosides / pharmacology*
  • HEK293 Cells
  • Humans
  • Insulin / metabolism
  • Insulin Secretion
  • Insulin-Secreting Cells / drug effects*
  • Insulin-Secreting Cells / metabolism
  • Male
  • Mice
  • Mice, Knockout
  • Patch-Clamp Techniques
  • Sweetening Agents / pharmacology*
  • TRPM Cation Channels / drug effects*
  • TRPM Cation Channels / metabolism
  • Taste / drug effects*

Substances

  • Blood Glucose
  • Diterpenes, Kaurane
  • Glucosides
  • Insulin
  • Sweetening Agents
  • TRPM Cation Channels
  • TRPM4 protein, human
  • TRPM5 protein, human
  • Trpm5 protein, mouse
  • stevioside
  • steviol
  • rebaudioside A