A soluble CD4 protein selectively inhibits HIV replication and syncytium formation

Nature. 1988 Jan 7;331(6151):78-81. doi: 10.1038/331078a0.

Abstract

The CD4 (T4) molecule is expressed on a subset of T lymphocytes involved in class II MHC recognition, and is probably the physiological receptor for one or more monomorphic regions of class II MHC (refs 1-3). CD4 also functions as a receptor for the human immunodeficiency virus (HIV) exterior envelope glycoprotein (gp120) (refs 4-9), being essential for virus entry into the host cell and for membrane fusion, which contributes to cell-to-cell transmission of the virus and to its cytopathic effects. We have used a baculovirus expression system to generate mg quantities of a hydrophilic extracellular segment of CD4. Concentrations of soluble CD4 in the nanomolar range, like certain anti-CD4 monoclonal antibodies, inhibit syncytium formation and HIV infection by binding gp120-expressing cells. Perhaps more importantly, class II specific T-cell interactions are uninhibited by soluble CD4 protein, whereas they are virtually abrogated by equivalent amounts of anti-T4 antibody. This may reflect substantial differences in CD4 affinity for gp120 and class II MHC.

MeSH terms

  • Animals
  • Antigens, Differentiation, T-Lymphocyte / metabolism*
  • Binding, Competitive
  • Cell Fusion*
  • Cell Line
  • Cricetinae
  • Cricetulus
  • Female
  • Fibroblasts / metabolism
  • HIV / physiology*
  • HIV Envelope Protein gp120
  • Humans
  • Ovary
  • Receptors, HIV
  • Receptors, Virus / metabolism*
  • Recombinant Fusion Proteins / metabolism
  • Recombinant Fusion Proteins / pharmacology*
  • Recombinant Proteins / pharmacology*
  • Retroviridae Proteins / metabolism
  • Solubility
  • T-Lymphocytes / metabolism
  • Virus Replication*

Substances

  • Antigens, Differentiation, T-Lymphocyte
  • HIV Envelope Protein gp120
  • Receptors, HIV
  • Receptors, Virus
  • Recombinant Fusion Proteins
  • Recombinant Proteins
  • Retroviridae Proteins