Potent neutralization of hepatitis A virus reveals a receptor mimic mechanism and the receptor recognition site

Proc Natl Acad Sci U S A. 2017 Jan 24;114(4):770-775. doi: 10.1073/pnas.1616502114. Epub 2017 Jan 10.

Abstract

Hepatitis A virus (HAV) infects ∼1.4 million people annually and, although there is a vaccine, there are no licensed therapeutic drugs. HAV is unusually stable (making disinfection problematic) and little is known of how it enters cells and releases its RNA. Here we report a potent HAV-specific monoclonal antibody, R10, which neutralizes HAV infection by blocking attachment to the host cell. High-resolution cryo-EM structures of HAV full and empty particles and of the complex of HAV with R10 Fab reveal the atomic details of antibody binding and point to a receptor recognition site at the pentamer interface. These results, together with our observation that the R10 Fab destabilizes the capsid, suggest the use of a receptor mimic mechanism to neutralize virus infection, providing new opportunities for therapeutic intervention.

Keywords: entry; neutralizing mechanism; picornavirus; receptor recognition; uncoating.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Antibodies, Monoclonal / immunology
  • Antibodies, Neutralizing / immunology*
  • Binding Sites / immunology
  • Capsid / immunology
  • Capsid Proteins / immunology
  • Female
  • Hepatitis A virus / immunology*
  • Humans
  • Immunoglobulin Fab Fragments / immunology
  • Mice
  • Mice, Inbred BALB C

Substances

  • Antibodies, Monoclonal
  • Antibodies, Neutralizing
  • Capsid Proteins
  • Immunoglobulin Fab Fragments

Associated data

  • PDB/5WTF
  • PDB/5WTE
  • PDB/5WTG
  • PDB/5WTH