Characterizing and targeting PDGFRA alterations in pediatric high-grade glioma

Oncotarget. 2016 Oct 4;7(40):65696-65706. doi: 10.18632/oncotarget.11602.

Abstract

Pediatric high-grade glioma (HGG, WHO Grade III and IV) is a devastating brain tumor with a median survival of less than two years. PDGFRA is frequently mutated/ amplified in pediatric HGG, but the significance of this finding has not been fully characterized. We hypothesize that alterations of PDGFRA will promote distinct prognostic and treatment implications in pediatric HGG. In order to characterize the impact of PDGFR pathway alterations, we integrated genomic data from pediatric HGG patients (n=290) from multiple pediatric datasets and sequencing platforms. Integration of multiple human datasets showed that PDGFRA mutation, but not amplification, was associated with older age in pediatric HGG (P= <0.0001). In multivariate analysis, PDGFRA mutation was correlated with worse prognosis (P = 0.026), while PDGFRA amplification was not (P = 0.11). By Kaplan-Meier analysis, non-brainstem HGG with PDGFRA amplification carried a worse prognosis than non-brainstem HGG without PDGFRA amplification (P = 0.021). There were no pediatric patients with PDGFRA-amplified HGG that survived longer than two years. Additionally, we performed paired molecular profiling (germline / tumor / primary cell culture) and targeting of an infant thalamic HGG with amplification and outlier increased expression of PDGFRA. Dasatinib inhibited proliferation most effectively. In summary, integration of the largest genomic dataset of pediatric HGG to date, allowed us to highlight that PDGFRA mutation is found in older pediatric patients and that PDGFRA amplification is prognostic in non-brainstem HGG. Future precision-medicine based clinical trials for pediatric patients with PDGFRA-altered HGG should consider the optimized delivery of dasatinib.

Keywords: PDGFRA amplification; PDGFRA mutation; brain tumor; pediatric high-grade glioma; tyrosine kinase inhibitor.

MeSH terms

  • Adolescent
  • Adult
  • Age Factors
  • Antineoplastic Agents / pharmacology
  • Apoptosis / drug effects
  • Biomarkers, Tumor / genetics*
  • Brain Neoplasms / drug therapy
  • Brain Neoplasms / genetics*
  • Brain Neoplasms / pathology
  • Cell Proliferation / drug effects
  • Child
  • Child, Preschool
  • Female
  • Follow-Up Studies
  • Gene Amplification*
  • Glioma / drug therapy
  • Glioma / genetics*
  • Glioma / pathology
  • Humans
  • Infant
  • Male
  • Mutation*
  • Neoplasm Grading
  • Receptor, Platelet-Derived Growth Factor alpha / genetics*
  • Survival Rate
  • Tumor Cells, Cultured
  • Young Adult

Substances

  • Antineoplastic Agents
  • Biomarkers, Tumor
  • Receptor, Platelet-Derived Growth Factor alpha